BDBM50339683 4-(Thiophen-3-yl)-N-(4-(4-(2-(2-fluoroethoxy)phenyl)piperazin-1-yl)-trans-but-2-enyl)benzamides oxalic acid salt::CHEMBL1689012
SMILES FCCOc1ccccc1N1CCN(C\C=C\CNC(=O)c2ccc(cc2)-c2ccsc2)CC1
InChI Key InChIKey=HFGAWEJFDVAEEA-ONEGZZNKSA-N
Data 5 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50339683
Affinity DataKi: 1.10nMAssay Description:Displacement of [125I]-IABN from human D3 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 70.5nMAssay Description:Displacement of [125I]-IABN from human D2 receptor transfected in human HEK 293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 182nMAssay Description:Binding affinity to human D4 receptor transfected in human HEK293 cells by gamma-countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.32E+3nMAssay Description:Displacement of [3H]-DTG from rat sigma2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 7.78E+3nMAssay Description:Displacement of [3H]-pentazocine from guinea pig sigma1 receptor by liquid scintillation countingMore data for this Ligand-Target Pair