BDBM50356013 CHEMBL1911374::CHEMBL1911375
SMILES FC(F)(F)c1ccc(Cn2nc3c(-c4ccncc4)c(cnn3c2=O)-c2ccc(Cl)cc2)cn1
InChI Key InChIKey=LOLQZUDLOOHVCH-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 7 hits for monomerid = 50356013
Affinity DataKi: 12nMAssay Description:Binding affinity to human CB1 receptor expressed in CHO cells by radioligand displacement based scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKd: 3.95nMAssay Description:Binding affinity to human CB1 receptor expressed in CHO cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 12.4nMAssay Description:Displacement of [3H]-SR-141716 from rat CB1 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 4.60nMAssay Description:Displacement of [3H]-SR-141716 from human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Displacement of [3H]BMS-725519 from rat brain CB1 receptor after 90 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKd: 29.1nMAssay Description:Binding affinity to rat brain CB1 receptor after 90 mins by scintillation countingMore data for this Ligand-Target Pair