BDBM50376902 CHEMBL408194
SMILES COC1=CC(=N\C1=C/c1[nH]c(C)cc1C)c1cc2ccccc2[nH]1
InChI Key InChIKey=RFTSSZJZXOSICM-GRSHGNNSSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 17 hits for monomerid = 50376902
Affinity DataKi: 1.00E+3nMAssay Description:Inhibition of BH3 peptide binding to human recombinant BCL-b by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Inhibition of BH3 peptide binding to human recombinant BCL-XL by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Mcgill University
Curated by ChEMBL
Mcgill University
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Inhibition of BH3 peptide binding to human recombinant MCL1 by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Inhibition of BH3 peptide binding to human recombinant BCL-w by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Inhibition of BH3 peptide binding to human recombinant A1 by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.11E+3nMAssay Description:Inhibition of Bcl2 (unknown origin)More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Mcgill University
Curated by ChEMBL
Mcgill University
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:Inhibition of MCl-1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 4.69E+3nMAssay Description:Inhibition of Bcl-xL (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 5.00E+3nMAssay Description:Inhibition of adenosine receptor A1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 7.01E+3nMAssay Description:Inhibition of Bcl-w (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.11E+3nMAssay Description:Inhibition of Bcl-2 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.69E+3nMAssay Description:Inhibition of monkey plasma renin activityMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Mcgill University
Curated by ChEMBL
Mcgill University
Curated by ChEMBL
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of Mcl-1 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Mcgill University
Curated by ChEMBL
Mcgill University
Curated by ChEMBL
Affinity DataEC50: 500nMAssay Description:Inhibition of GST-tagged recombinant Mcl1 interaction with biotinylated Bim peptide by ELISA based competitive binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 600nMAssay Description:Inhibition of GST-tagged recombinant Bfl1 interaction with biotinylated Bim peptide by ELISA based competitive binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 900nMAssay Description:Inhibition of GST-tagged recombinant Bcl-XL interaction with biotinylated Bim peptide by ELISA based competitive binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 300nMAssay Description:Inhibition of GST-tagged recombinant Bcl2 interaction with biotinylated Bim peptide by ELISA based competitive binding assayMore data for this Ligand-Target Pair