BDBM50380620 CHEMBL2016866
SMILES NC(=N)c1ccc(CNC(=O)[C@@H]2CCC(=O)NCc3cccc(CNC(=O)CC[C@@H](NS(=O)(=O)Cc4ccccc4)C(=O)N2)c3)cc1
InChI Key InChIKey=DBLYNSSCIKMVDW-WUFINQPMSA-N
Data 9 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 9 hits for monomerid = 50380620
TargetVitamin K-dependent protein C(Homo sapiens (Human))
Philipps University Marburg
Curated by ChEMBL
Philipps University Marburg
Curated by ChEMBL
Affinity DataKi: 5.10nMAssay Description:Inhibition of activated protein C by dixon plot methodMore data for this Ligand-Target Pair
Affinity DataKi: 25nMpH: 8.0Assay Description:The inhibition constants for human plasmin (h plasmin), human plasma kallikrein (h PK), thrombin and factor Xa were determined in analogy to a previo...More data for this Ligand-Target Pair
Affinity DataKi: 25.4nMAssay Description:Inhibition of plasma kallikrein by dixon plot methodMore data for this Ligand-Target Pair
Affinity DataKi: 431nMpH: 8.0Assay Description:The inhibition constants for human plasmin (h plasmin), human plasma kallikrein (h PK), thrombin and factor Xa were determined in analogy to a previo...More data for this Ligand-Target Pair
Affinity DataKi: 431nMAssay Description:Inhibition of plasmin by dixon plot methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.02E+3nMpH: 8.0Assay Description:The inhibition constants for human plasmin (h plasmin), human plasma kallikrein (h PK), thrombin and factor Xa were determined in analogy to a previo...More data for this Ligand-Target Pair
Affinity DataKi: 2.02E+3nMAssay Description:Inhibition of thrombin by dixon plot methodMore data for this Ligand-Target Pair
Affinity DataKi: 3.43E+3nMAssay Description:Inhibition of factor 10a by dixon plot methodMore data for this Ligand-Target Pair
Affinity DataKi: 3.43E+3nMpH: 8.0Assay Description:The inhibition constants for human plasmin (h plasmin), human plasma kallikrein (h PK), thrombin and factor Xa were determined in analogy to a previo...More data for this Ligand-Target Pair