BDBM50391482 CHEMBL2147218

SMILES Cc1ncc(cn1)-c1ccccc1CCNC(=O)c1cnc(OCCOCC(F)(F)F)c(C)c1

InChI Key InChIKey=DZZDGFAFADZZQZ-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50391482   

TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50391482(CHEMBL2147218)
Affinity DataIC50: <3.16E+4nMAssay Description:Inhibition of human Nav1.5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50391482(CHEMBL2147218)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells by whole cell voltage-clamp electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed