BDBM50400541 CHEMBL2204950
SMILES COc1cccc(CNC(=O)N[C@@H](CC(C)C)C(=O)NO)c1
InChI Key InChIKey=VRQZXSUCWGBJIY-ZDUSSCGKSA-N
Data 4 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50400541
Affinity DataIC50: 290nMAssay Description:Inhibition of APN in porcine kidney microsome assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substra...More data for this Ligand-Target Pair
Affinity DataIC50: 790nMAssay Description:Inhibition of APN in human ES2 cell surface assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substrate...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of recombinant MMP-2 using succinylated gelatin as substrate incubated for 10 mins before addition of substrate measured after 60 mins by ...More data for this Ligand-Target Pair
Affinity DataIC50: 5.61E+3nMAssay Description:Inhibition of mouse APNMore data for this Ligand-Target Pair