BDBM50400772 CHEMBL2204985

SMILES CCc1cnc(nc1)N1CCC(CC1)n1ncc(COc2ccc(cc2F)C#N)c1C#N

InChI Key InChIKey=SFWORIUDBFNINU-UHFFFAOYSA-N

Data  1 KI  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50400772   

TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400772(CHEMBL2204985)
Affinity DataKi:  9.30nMAssay Description:Binding affinity to human GPR119More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400772(CHEMBL2204985)
Affinity DataEC50:  2.80nMAssay Description:Agonist activity at GPR119 in human HEK293 cells assessed as cAMP level by beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400772(CHEMBL2204985)
Affinity DataEC50:  5.40nMAssay Description:Agonist activity at GPR119 in human U20S cells assessed as binding to beta-arrestin by chemilumiscence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed