BDBM50415643 CHEMBL1078642::UR-PI376
SMILES N#CNC(NCCSc1ccccc1)=NCCCCc1cnc[nH]1
InChI Key InChIKey=DHHDEHNHEBYRPQ-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 7 hits for monomerid = 50415643
Affinity DataKi: 57.5nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 525nMAssay Description:Displacement of [3H]N-alpah-methylhistamine from human histamine H3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.07E+3nMAssay Description:Displacement of [3H]tiotidine from human histamine H2 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.57E+4nMAssay Description:Displacement of [3H]mepyramine from human histamine H1 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 33.9nMAssay Description:Agonist activity at human histamine H4 receptor expressed in Sf9 cells coexpressing RGS19 protein by steady-state GTPase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 720nMAssay Description:Agonist activity at human histamine H3 receptor expressed in sf9 cell membrane co-expressing mammalian Galphai2 and Gbeta1gamma2 incubated for 90 min...More data for this Ligand-Target Pair
Affinity DataEC50: 37nMAssay Description:Agonist activity at human histamine H4 receptor expressed in sf9 cell membrane co-expressing mammalian Galphai2 and Gbeta1gamma2 incubated for 90 min...More data for this Ligand-Target Pair