BDBM50415761 CHEMBL5285102
SMILES Fc1ccc(CN2CCN(CC2)C(=O)\C=C\c2ccccc2Cl)cc1
InChI Key InChIKey=RMDYFILMTQCLCQ-JXMROGBWSA-N
Data 5 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50415761
Affinity DataIC50: 5nMAssay Description:Displacement of [3H]UR-MK299 from human neuropeptide Y Y2 receptor expressed in CHO cells measured after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Agonist activity at human neuropeptide Y Y4 receptor expressed in HEK293T cells co-expressing CRE-controlled gene reporter firefly luciferase assesse...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human GAL4-fused RORbeta LBD transfected in HEK293T cell measured for 16 to 20 hrs by by dual-glo luciferase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.54E+3nMAssay Description:Inhibition of human GAL4-fused RORalpha LBD transfected in HEK293T cell measured for 16 to 20 hrs by by dual-glo luciferase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 42nMAssay Description:Inhibition of human GAL4-fused RORgammat LBD transfected in HEK293T cell measured for 16 to 20 hrs by by dual-glo luciferase assayMore data for this Ligand-Target Pair