BDBM50426570 CHEMBL2324344
SMILES CCCC(=O)C1CCN(CC1)c1ncnc2CCN(Cc12)C(=O)c1ccc(cc1)-c1ccccc1
InChI Key InChIKey=CJZGRIRZVHNUSM-UHFFFAOYSA-N
Data 7 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 7 hits for monomerid = 50426570
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
University Of Kansas Specialized Chemistry Center
Curated by ChEMBL
University Of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of TASK-1 (unknown origin) expressed in CHO cells by thallium flux assayMore data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Inhibition of TASK-3 (unknown origin)More data for this Ligand-Target Pair
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
University Of Kansas Specialized Chemistry Center
Curated by ChEMBL
University Of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of TASK-1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Inhibition of human TASK3 expressed in HEK293 cells by Qpatch HT platform based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 243nMAssay Description:Inhibition of human TASK3 expressed in Xenopus oocytes by whole cell voltage clamp assayMore data for this Ligand-Target Pair
TargetPotassium channel subfamily K member 9(Rattus norvegicus)
Universidad De Talca
Curated by ChEMBL
Universidad De Talca
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of rat TASK3 expressed in (FRT) epithelial cells by chamber based electrophysiology assayMore data for this Ligand-Target Pair
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
University Of Kansas Specialized Chemistry Center
Curated by ChEMBL
University Of Kansas Specialized Chemistry Center
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of human TASK1 expressed in HEK293 cells by Qpatch HT platform based assayMore data for this Ligand-Target Pair