BDBM50432950 CHEMBL2377735

SMILES O=C(Nc1nc2ccccc2s1)N(CCC(c1ccccc1)c1ccccc1)CCN1CCOCC1

InChI Key InChIKey=GCEKXNZJEPZBBC-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50432950   

TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432950(CHEMBL2377735)
Affinity DataEC50:  20nMAssay Description:Positive allosteric modulation of human CaSR expressed in CHO cells assessed as increase in intracellular calcium level after 5 hrs by luciferase rep...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed