BDBM50439188 CHEMBL2418791::US9126987, 7
SMILES C=CCSc1nnc(o1)-c1ccc2[nH]cnc2c1
InChI Key InChIKey=XVIDYGSAQLUXTC-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50439188
Affinity DataKi: 5.26E+3nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Escherichia coli DH5alpha using H-Gln-AMC as substrate by fluorometric analysis in presence of py...More data for this Ligand-Target Pair
Affinity DataKi: 5.26E+3nM ΔG°: -7.32kcal/mole IC50: 7.23E+3nMpH: 8.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30 C. QC activity was evaluated fluorometricall...More data for this Ligand-Target Pair
Affinity DataIC50: 7.23E+3nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Escherichia coli DH5alpha using H-Gln-AMC as substrate by fluorometric analysis in presence of py...More data for this Ligand-Target Pair