BDBM50458583 CHEMBL4205609

SMILES COc1cccc(c1)C(=O)c1ccc2n(ccc2c1)S(=O)(=O)c1cccc(\C=C\C(=O)NO)c1

InChI Key InChIKey=MPHCHZFSBARRJN-DHZHZOJOSA-N

Data  6 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50458583   

TargetPolyamine deacetylase HDAC10(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50458583(CHEMBL4205609)
Affinity DataIC50:  7.74E+3nMAssay Description:Displacement of [3H]glycine from GlyT2 in Wistar rat brainstem cells after 10 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50458583(CHEMBL4205609)
Affinity DataIC50:  1.21E+3nMAssay Description:Inhibition of human HDAC1 using RHKKAc peptide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50458583(CHEMBL4205609)
Affinity DataIC50:  1.81E+3nMAssay Description:Inhibition of human HDAC6 using RHKKAc peptide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50458583(CHEMBL4205609)
Affinity DataIC50:  323nMAssay Description:Inhibition of human HDAC3 using RHKKAc peptide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50458583(CHEMBL4205609)
Affinity DataIC50:  3.53E+3nMAssay Description:Inhibition of human HDAC8 using RHKAcKAc peptide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50458583(CHEMBL4205609)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of human HDAC2 using RHKKAc peptide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed