BDBM50463108 CHEMBL4244874

SMILES CCn1c2ccccc2c2cc(NC(=O)N3CCC(CC3)C(C)=O)ccc12

InChI Key InChIKey=DZRSNKIGPLOVQE-UHFFFAOYSA-N

Data  1 KI  1 IC50  1 Kd

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50463108   

TargetDNA repair protein REV1(Homo sapiens)
University Of Connecticut

Curated by ChEMBL
LigandPNGBDBM50463108(CHEMBL4244874)
Affinity DataKi:  8.90E+3nMAssay Description:Displacement of FAM-labelled polkappa-RIR peptide from recombinant human C-terminal Rev1 (1158 to 1251 residues) expressed in Escherichia coli BL21(D...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA repair protein REV1(Homo sapiens)
University Of Connecticut

Curated by ChEMBL
LigandPNGBDBM50463108(CHEMBL4244874)
Affinity DataKd:  6.90E+3nMAssay Description:Displacement of FAM-labelled polkappa-RIR peptide from recombinant human C-terminal Rev1 (1158 to 1251 residues) expressed in Escherichia coli BL21(D...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA repair protein REV1(Homo sapiens)
University Of Connecticut

Curated by ChEMBL
LigandPNGBDBM50463108(CHEMBL4244874)
Affinity DataIC50:  4.60E+3nMAssay Description:Displacement of FAM-labelled polkappa-RIR peptide from recombinant human C-terminal Rev1 (1158 to 1251 residues) expressed in Escherichia coli BL21(D...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed