BDBM50470544 CHEMBL4282765
SMILES CC(C)[C@H](NC(=O)[C@@H](NC(=O)[C@@H]1OC(=O)[C@H]1C(C)C)C(C)C)C(O)=O
InChI Key InChIKey=PDPYJYDVMZXUKQ-ZDEQEGDKSA-N
Data 4 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50470544
TargetmRNA cap guanine-N7 methyltransferase(Homo sapiens)
New Mexico Institute Of Mining And Technology
Curated by ChEMBL
New Mexico Institute Of Mining And Technology
Curated by ChEMBL
Affinity DataIC50: 6.16E+4nMAssay Description:Inhibition of yeast 20S proteasome beta2 subunit using SUC-RLR-AMC as substrate pretreated for 30 mins followed by substrate addition and measured af...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
New Mexico Institute Of Mining And Technology
Curated by ChEMBL
New Mexico Institute Of Mining And Technology
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Inhibition of 20S proteasome beta5 subunit in human Jurkat cell lysate using Suc-LLVY-AMC as substrate pretreated for 30 mins followed by substrate a...More data for this Ligand-Target Pair
TargetmRNA cap guanine-N7 methyltransferase(Homo sapiens)
New Mexico Institute Of Mining And Technology
Curated by ChEMBL
New Mexico Institute Of Mining And Technology
Curated by ChEMBL
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of yeast 20S proteasome beta1 subunit using fluorescent substrate pretreated for 30 mins followed by substrate addition and measured after...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-8(Homo sapiens (Human))
New Mexico Institute Of Mining And Technology
Curated by ChEMBL
New Mexico Institute Of Mining And Technology
Curated by ChEMBL
Affinity DataIC50: 681nMAssay Description:Inhibition of human immunoproteasome beta5 subunit using Suc-RLR-AMC as substrate pretreated for 30 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair