BDBM50470559 CHEMBL4285979
SMILES [H][C@]1([C@@H](C)CC)[C@@H](OC1=O)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](C(C)C)C(=O)OCC=C
InChI Key InChIKey=HCQRRPYERGCDMA-QUSNUVHPSA-N
Data 4 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50470559
TargetProteasome subunit beta type-8(Homo sapiens (Human))
New Mexico Institute Of Mining And Technology
Curated by ChEMBL
New Mexico Institute Of Mining And Technology
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of human immunoproteasome beta5 subunit using Suc-RLR-AMC as substrate pretreated for 30 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
New Mexico Institute Of Mining And Technology
Curated by ChEMBL
New Mexico Institute Of Mining And Technology
Curated by ChEMBL
Affinity DataIC50: 9.40nMAssay Description:Inhibition of 20S proteasome beta5 subunit in human Jurkat cell lysate using Suc-LLVY-AMC as substrate pretreated for 30 mins followed by substrate a...More data for this Ligand-Target Pair
TargetmRNA cap guanine-N7 methyltransferase(Homo sapiens)
New Mexico Institute Of Mining And Technology
Curated by ChEMBL
New Mexico Institute Of Mining And Technology
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of yeast 20S proteasome beta2 subunit using SUC-RLR-AMC as substrate pretreated for 30 mins followed by substrate addition and measured af...More data for this Ligand-Target Pair
TargetmRNA cap guanine-N7 methyltransferase(Homo sapiens)
New Mexico Institute Of Mining And Technology
Curated by ChEMBL
New Mexico Institute Of Mining And Technology
Curated by ChEMBL
Affinity DataIC50: 779nMAssay Description:Inhibition of yeast 20S proteasome beta1 subunit using fluorescent substrate pretreated for 30 mins followed by substrate addition and measured after...More data for this Ligand-Target Pair