BDBM50504145 CHEMBL1711265
SMILES Cc1ccccc1C(=O)NCC(=O)Nc1ccc(C)c(c1)S(=O)(=O)N1CCCCCC1
InChI Key InChIKey=AQTOEFKBMJNVRD-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50504145
Affinity DataIC50: 1.26E+4nMAssay Description:Displacement of SGRG-K(Ac)-GG-K(Ac)-GLG-K(Ac)-GGAKRHRKV-biotin) from His6/FLAG-tagged TEV fused ATAD2 bromodomain (981 to 1121 residues) (unknown ori...More data for this Ligand-Target Pair
Affinity DataKd: 3.16E+4nMAssay Description:Binding affinity to His6/FLAG-tagged TEV fused ATAD2 bromodomain (950 to 1148 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cell...More data for this Ligand-Target Pair
Affinity DataIC50: 3.98E+4nMAssay Description:Inhibition of ATAD2 bromodomain in human HUT78 chromatin lysate after 2 hrs by bromosphere competition binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: <5.01E+4nMAssay Description:Displacement of Alexa Fluor 647 labelled ligand from His6-tagged BRD4 BD2 (1 to 477 residues)/BD1 Y97A mutant (unknown origin) after 30 mins by TR-FR...More data for this Ligand-Target Pair
Affinity DataIC50: <5.01E+4nMAssay Description:Displacement of Alexa Fluor 647 labelled ligand from His6-tagged BRD4 BD1 (1 to 477 residues)/BD2 Y390A mutant (unknown origin) after 30 mins by TR-F...More data for this Ligand-Target Pair