BDBM50508743 CHEMBL4460141
SMILES CC(=O)Nc1ncc(CN2CCC3(CCN(C3)c3ncc(C)cc3C)C2)s1
InChI Key InChIKey=RROPSOUKMJSJQR-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50508743
Affinity DataIC50: 209nMAssay Description:Inhibition of OGA in HEK293 cells assessed as increase in O-GlcNAcylated protein level by Hoechst staining based microscopic methodMore data for this Ligand-Target Pair
Affinity DataIC50: 3.90nMAssay Description:Inhibition of recombinant human full length OGA using FM-GlcNAc as substrate preincubated for 60 mins followed by substrate addition and measured aft...More data for this Ligand-Target Pair