BDBM50512959 CHEMBL4454766
SMILES CCCCc1ccc(cc1)[C@H]1C[C@H](CN(C)C1)Nc1nc2cc[nH]c2c(=O)n1C
InChI Key InChIKey=UQXYUSOVVAUCIZ-RBUKOAKNSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50512959
Affinity DataKd: 183nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Inhibition of biotinylated peptide binding to human GST-tagged PCAF bromodomain expressed in Escherichia coli Rosetta (DE3) measured after 15 hrs by ...More data for this Ligand-Target Pair