BDBM50512979 CHEMBL4457684
SMILES CN1C[C@@H](C[C@@H](C1)c1ccc2ccccc2c1)Nc1nc2cc[nH]c2c(=O)n1C
InChI Key InChIKey=ZAJOVXHUHHARKS-RBUKOAKNSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50512979
Affinity DataKd: 103nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataIC50: 47nMAssay Description:Inhibition of biotinylated peptide binding to human GST-tagged PCAF bromodomain expressed in Escherichia coli Rosetta (DE3) measured after 15 hrs by ...More data for this Ligand-Target Pair