BDBM50520571 CHEMBL4447794
SMILES CN(c1cccc(CNc2nc(Nc3ccc(OCCOCCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCc4ccc(cc4)-c4scnc4C)C(C)(C)C)cc3)ncc2C(F)(F)F)c1)S(C)(=O)=O
InChI Key InChIKey=MVULIYLBRNHLEE-LFHXYJAASA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50520571
Affinity DataIC50: 6.5nMAssay Description:Inhibition of human recombinant FAK using poly[Glu:Tyr] (4:1) substrate in presence of 10 mM ATP and [gamma33P]-ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 6.5nMAssay Description:Inhibition of FAK (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Induction of degradation of Fak in human PC-3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of human FAK using poly (Glu,Tyr) as substrate by radiometric HotSpot kinase assayMore data for this Ligand-Target Pair