BDBM50528924 CHEMBL4473519
SMILES NC(=O)c1ccn(c1)-c1cccc(OC(=O)NCCN2CCN(CC2)c2ccccc2)c1
InChI Key InChIKey=WGOUWABLRGOCPZ-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 8 hits for monomerid = 50528924
Affinity DataKi: 16nMAssay Description:Inhibition of FAAH in mouse brain membranes assessed as inhibitory constant using [14C]-AEA as substrate incubated for 15 mins by scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 105nMAssay Description:Displacement of [3H]-spiperone from human D3 receptor expressed in CHO cells co-expressing Galpha16 incubated for 120 mins by liquid scintillation co...More data for this Ligand-Target Pair
Affinity DataKi: 105nMAssay Description:Displacement of [3H]-spiperone from human D3 receptor expressed in CHO cells co-expressing Galpha16 incubated for 120 mins by liquid scintillation co...More data for this Ligand-Target Pair
Affinity DataKi: 186nMAssay Description:Displacement of [3H]-spiperone from human D2 receptor expressed in CHO cells co-expressing Galpha16 incubated for 120 mins by liquid scintillation co...More data for this Ligand-Target Pair
Affinity DataKi: 186nMAssay Description:Displacement of [3H]-spiperone from human D2 receptor expressed in CHO cells co-expressing Galpha16 incubated for 120 mins by liquid scintillation co...More data for this Ligand-Target Pair
Affinity DataIC50: 58nMAssay Description:Inhibition of FAAH in mouse brain membranes using [14C]-AEA as substrate incubated for 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Siena
Curated by ChEMBL
University Of Siena
Curated by ChEMBL
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells incubated for 72 hrs by patch clamp assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Siena
Curated by ChEMBL
University Of Siena
Curated by ChEMBL
Affinity DataIC50: 5.25E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells incubated for 72 hrs by patch clamp assayMore data for this Ligand-Target Pair