BDBM50551201 CHEMBL4761556
SMILES [H][C@@]1(CC[C@@]2([H])[C@]3([H])CC[C@]4([H])C[C@@H](CC[C@]4(C)[C@@]3([H])CC[C@]12C)OC(=O)NCC)[C@H](C)CCC(=O)N[C@H](CC(O)=O)Cc1c[nH]c2ccccc12
InChI Key InChIKey=JZDJKWCLKGBXIC-LRVDEVEJSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 15 hits for monomerid = 50551201
Affinity DataKi: 300nMAssay Description:Competitive inhibition of biotinylated ephrin-A1-Fc binding to EphA2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Displacement of biotinylated ephrin-B1-Fc from mouse EphB6 Fc preincubated for 1 hr followed by ephrin-B1-FC addition and measured after 4 hrs by ELI...More data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+4nMAssay Description:Displacement of biotinylated ephrin-B1-Fc from mouse EphB3 Fc preincubated for 1 hr followed by ephrin-B1-FC addition and measured after 4 hrs by ELI...More data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Displacement of biotinylated ephrin-A1-Fc from human EphA1 Fc preincubated for 1 hr followed by ephrin-A1-FC addition and measured after 4 hrs by ELI...More data for this Ligand-Target Pair
Affinity DataIC50: 4.50E+3nMAssay Description:Displacement of biotinylated ephrin-A1-Fc from mouse EphA3 Fc preincubated for 1 hr followed by ephrin-A1-FC addition and measured after 4 hrs by ELI...More data for this Ligand-Target Pair
Affinity DataIC50: 6.40E+3nMAssay Description:Displacement of biotinylated ephrin-A1-Fc from mouse EphA4 Fc preincubated for 1 hr followed by ephrin-A1-FC addition and measured after 4 hrs by ELI...More data for this Ligand-Target Pair
Affinity DataIC50: 4.40E+3nMAssay Description:Displacement of biotinylated ephrin-A1-Fc from rat EphA5 Fc preincubated for 1 hr followed by ephrin-A1-FC addition and measured after 4 hrs by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+4nMAssay Description:Displacement of biotinylated ephrin-A1-Fc from mouse EphA6 Fc preincubated for 1 hr followed by ephrin-A1-FC addition and measured after 4 hrs by ELI...More data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Displacement of biotinylated ephrin-A1-Fc from mouse EphA7 Fc preincubated for 1 hr followed by ephrin-A1-FC addition and measured after 4 hrs by ELI...More data for this Ligand-Target Pair
Affinity DataIC50: 7.70E+3nMAssay Description:Displacement of biotinylated ephrin-A1-Fc from mouse EphA8 Fc preincubated for 1 hr followed by ephrin-A1-FC addition and measured after 4 hrs by ELI...More data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+4nMAssay Description:Displacement of biotinylated ephrin-B1-Fc from mouse EphB2 Fc preincubated for 1 hr followed by ephrin-B1-FC addition and measured after 4 hrs by ELI...More data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Displacement of biotinylated ephrin-B1-Fc from rat EphB1 Fc preincubated for 1 hr followed by ephrin-B1-FC addition and measured after 4 hrs by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Displacement of biotinylated ephrin-B1-Fc from mouse EphB4 Fc preincubated for 1 hr followed by ephrin-B1-FC addition and measured after 4 hrs by ELI...More data for this Ligand-Target Pair
Affinity DataIC50: 950nMAssay Description:Displacement of biotinylated ephrin-A1-Fc from recombinant mouse c-terminal His6-tagged EphA2 Fc (Ala22 to Ala535 residues) preincubated for 1 hr fol...More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Antagonist activity at EphA2-Fc in human PC3 cells assessed as reduction in ephrin-A1-Fc stimulated EphA2 phosphorylation preincubated for 20 mins fo...More data for this Ligand-Target Pair