BDBM50569995 CHEMBL4874284
SMILES CCS(=O)(=O)c1ccc(CNC(=O)c2ccc(CCN3CCOc4ccc(OC(C)C)cc34)cc2)nc1
InChI Key InChIKey=PGCXGBWVFHQCIO-UHFFFAOYSA-N
Data 2 EC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50569995
Affinity DataEC50: 4.60nMAssay Description:Agonist activity at APC-labelled RORgammat (unknown origin) assessed as biotinylated SRC recruitment measured after 1 hr by dual FRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 135nMAssay Description:Agonist activity at human RORgammat LBD expressed in HEK293T cells assessed increase in Gal4 reporter gene transcription measured after 16 to 20 hrs ...More data for this Ligand-Target Pair