BDBM50574750 CHEMBL4850758
SMILES CC(C)(C)OC(=O)N[C@@H]1CCN(C1)C(c1ccc(cc1)-c1ccncc1)c1cc2OCOc2cc1O
InChI Key InChIKey=UMKHMAZNAYZVDJ-OSMGYRLQSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 7 hits for monomerid = 50574750
Affinity DataKi: 293nMAssay Description:Mixed inhibition of human KDM4D expressed in Escherichia coli BL21(DE3) using H3(1-21)K9me3 peptide and varying concentrations of 2-OG as substrate p...More data for this Ligand-Target Pair
Affinity DataKd: 36nMAssay Description:Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) assessed as equilibrium dissociation constant measured by isothermal titration cal...More data for this Ligand-Target Pair
Affinity DataIC50: 3.71E+4nMAssay Description:Inhibition of KDM6A (unknown origin) by AlphaLISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of KDM4A (unknown origin) by AlphaLISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of KDM5A (unknown origin) by AlphaLISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) using biotinylated H3-derived peptide and 2-OG as substrate preincubated for 15 mi...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of KDM3B (unknown origin) by AlphaLISA assayMore data for this Ligand-Target Pair