BDBM511431 (-)-(1 S,5R)-2-methyl-4-(5-(phenylethynyl)pyridin-2-yl)-2,4-diazabicyclo[3.2.0]heptan-3-one::US11059766, Example 1
SMILES CN1[C@H]2CC[C@H]2N(C1=O)c1ccc(cn1)C#Cc1ccccc1
InChI Key InChIKey=GUFIEMPVYLURJX-DLBZAZTESA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 511431
Affinity DataKi: 9nMAssay Description:For binding experiments, cDNA encoding human mGlu5a receptor was transiently transfected into EBNA cells using a procedure described by Schlaeger and...More data for this Ligand-Target Pair
Affinity DataEC50: 9nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu5a receptor was generated; for the work with mGlu5 Positive ...More data for this Ligand-Target Pair