BDBM518438 2-[4-[2-[(2S)-2-Methylazetidin-1-yl]-6- (trifluoromethyl)pyrimidin-4-yl]pyrazol- 1-yl]-1-[(2S)-2-methylpiperazin-1- yl]ethanone::US11124500, Example 30
SMILES C[C@H]1CCN1c1nc(cc(n1)C(F)(F)F)-c1cnn(CC(=O)N2CCNC[C@@H]2C)c1
InChI Key InChIKey=DPIAHCRTJNEWNS-STQMWFEESA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 518438
Affinity DataIC50: 57.8nMAssay Description:The intrinsic potency for inhibition of KHK C or A activity may be measured using an enzymatic assay which measures the production of FIP. Compounds ...More data for this Ligand-Target Pair
Affinity DataIC50: 46.3nMAssay Description:The intrinsic potency for inhibition of KHK C or A activity may be measured using an enzymatic assay which measures the production of FIP. Compounds ...More data for this Ligand-Target Pair