BDBM531994 N-[4-(2-Amino-5-{4-[(4-methylpiperazin-1-yl)methyl]phenyl}pyridin-3-yl)phenyl]-5-(4-methylphenyl)-4-oxo-1-(tetrahydro-2H-pyran-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide methanesulfonate::US11208403, Example 71
SMILES CN1CCN(Cc2ccc(cc2)-c2cnc(N)c(c2)-c2ccc(NC(=O)c3cn(CC4CCOCC4)cc(-c4ccc(C)cc4)c3=O)cc2)CC1
InChI Key InChIKey=IPHZKBACASVMHL-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 531994
Affinity DataIC50: 64nMAssay Description:A kinase dilution solution containing 20 ng/ml Mer (the 528th to 999th amino acids of the intracellular domain of human MER expressed as a fusion pro...More data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:A kinase dilution solution containing 170 ng/ml AXL (the 464th to 885th amino acids of the intracellular domain of human AXL expressed as a fusion pr...More data for this Ligand-Target Pair