BDBM532438 US11214548, Compound 634

SMILES CNC(=O)[C@@H](NC(=O)c1nn(c2[C@@H]3C[C@@H]3Cc12)-c1ccc(F)cc1F)C(C)(C)C

InChI Key InChIKey=WRFJHFSIGZXCCO-AJLCLMPTSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 532438   

TargetCannabinoid receptor 1(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM532438(US11214548, Compound 634)
Affinity DataEC50:  0.170nMAssay Description:Table D: Radioligand binding assays for human CB2 receptors were performed using two different agonist radioligands, [3H]CP55,940 and [3H]WIN55,212-2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCannabinoid receptor 2(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM532438(US11214548, Compound 634)
Affinity DataEC50:  1.10nMAssay Description:Table B: HTRF assay was carried out using a two-step protocol essentially according to the kit manufacturer's instructions, in 20 μL total v...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent