BDBM536862 (S)-1-(3-(6-(1-methyl-1H-pyrazol-4-yl)naphthalen-1-yl)-1-(tetrahydrofuran-3-yl)-6,7-dihydro-1H-pyrazolo[4,3-c]pyridin-5(4H)-yl)ethanone::US11247989, Example 36

SMILES CC(=O)N1CCc2c(C1)c(nn2[C@H]1CCOC1)-c1cccc2cc(ccc12)-c1cnn(C)c1

InChI Key InChIKey=FTAJMIWEBHWZEB-NRFANRHFSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 536862   

TargetCREB-binding protein(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM536862((S)-1-(3-(6-(1-methyl-1H-pyrazol-4-yl)naphthalen-1...)
Affinity DataIC50:  1.39nMAssay Description:His/Flag epitope tagged CBP was cloned, expressed, and purified to homogeneity. CBP binding and inhibition was assessed by monitoring the engagement ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent