BDBM536875 2-cyano-N-methyl-3-(3-(1-methyl-1H-pyrazol-4-yl)isoquinolin-8-yl)-1-(tetrahydro-2H-pyran-4-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridine-5(4H)-carboxamide::US11247989, Example 49
SMILES CNC(=O)N1CCc2c(C1)c(c(C#N)n2C1CCOCC1)-c1cccc2cc(ncc12)-c1cnn(C)c1
InChI Key InChIKey=FHDSEZXJVYUDBE-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 536875
Affinity DataIC50: 1.42nMAssay Description:His/Flag epitope tagged CBP was cloned, expressed, and purified to homogeneity. CBP binding and inhibition was assessed by monitoring the engagement ...More data for this Ligand-Target Pair