BDBM576049 4-(1-benzyl-2-methyl-1H- imidazo[4,5-b]pyridin-6-yl)-6- methyl-1H-pyrrolo[2,3-c] pyridin-7(6H)-one::US11466034, Example 6
SMILES Cc1nc2ncc(cc2n1Cc1ccccc1)-c1cn(C)c(=O)c2[nH]ccc12
InChI Key InChIKey=NTRXALHVKBFJRO-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 576049
TargetBromodomain-containing protein 4 [349-460](Homo sapiens (Human))
Betta Pharmaceuticals
US Patent
Betta Pharmaceuticals
US Patent
Affinity DataIC50: 2.80nMAssay Description:The assays of BRD4 (D1) and BRD4 (D2) were conducted in a 384-well polystyrene plate. The test compounds were first serially diluted in DMSO and the ...More data for this Ligand-Target Pair
Affinity DataIC50: 7.60nMAssay Description:The assays of BRD4 (D1) and BRD4 (D2) were conducted in a 384-well polystyrene plate. The test compounds were first serially diluted in DMSO and the ...More data for this Ligand-Target Pair