BDBM576051 6-methyl-4-(2-methyl-1H- imidazo[4,5-b]pyridin-6-yl)-1,6- dihydro-7H-pyrrolo[2,3-c] pyridin-7-one::US11466034, Example 8
SMILES Cc1nc2ncc(cc2[nH]1)-c1cn(C)c(=O)c2[nH]ccc12
InChI Key InChIKey=PIXIOGOVJJLZSH-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 576051
TargetBromodomain-containing protein 4 [349-460](Homo sapiens (Human))
Betta Pharmaceuticals
US Patent
Betta Pharmaceuticals
US Patent
Affinity DataIC50: 6nMAssay Description:The assays of BRD4 (D1) and BRD4 (D2) were conducted in a 384-well polystyrene plate. The test compounds were first serially diluted in DMSO and the ...More data for this Ligand-Target Pair
Affinity DataIC50: 39.9nMAssay Description:The assays of BRD4 (D1) and BRD4 (D2) were conducted in a 384-well polystyrene plate. The test compounds were first serially diluted in DMSO and the ...More data for this Ligand-Target Pair