BDBM576063 4-(1-(4-chlorobenzyl)-2-methyl- 1H-imidazo[4,5-b]pyrazin- 6-yl)-6-methyl-1H-pyrrolo [2,3-c]pyridin-7(6H)-one::US11466034, Example 18
SMILES Cc1nc2ncc(nc2n1Cc1ccc(Cl)cc1)-c1cn(C)c(=O)c2[nH]ccc12
InChI Key InChIKey=ZGLSYPGLUNRMHV-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 576063
TargetBromodomain-containing protein 4 [349-460](Homo sapiens (Human))
Betta Pharmaceuticals
US Patent
Betta Pharmaceuticals
US Patent
Affinity DataIC50: 1.70nMAssay Description:The assays of BRD4 (D1) and BRD4 (D2) were conducted in a 384-well polystyrene plate. The test compounds were first serially diluted in DMSO and the ...More data for this Ligand-Target Pair
Affinity DataIC50: 6.90nMAssay Description:The assays of BRD4 (D1) and BRD4 (D2) were conducted in a 384-well polystyrene plate. The test compounds were first serially diluted in DMSO and the ...More data for this Ligand-Target Pair