BDBM576066 4-(1-(1-(4-chlorophenyl)ethyl)- 2-methyl-1H-imidazo[4,5-b] pyrazin-6-yl)-6-methyl-1,6- dihydro-7H-pyrrolo[2,3-c] pyridin-7-one::US11466034, Example 21
SMILES CC(c1ccc(Cl)cc1)n1c(C)nc2ncc(nc12)-c1cn(C)c(=O)c2[nH]ccc12
InChI Key
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 576066
TargetBromodomain-containing protein 4 [349-460](Homo sapiens (Human))
Betta Pharmaceuticals
US Patent
Betta Pharmaceuticals
US Patent
Affinity DataIC50: 1.80nMAssay Description:The assays of BRD4 (D1) and BRD4 (D2) were conducted in a 384-well polystyrene plate. The test compounds were first serially diluted in DMSO and the ...More data for this Ligand-Target Pair
Affinity DataIC50: 6.10nMAssay Description:The assays of BRD4 (D1) and BRD4 (D2) were conducted in a 384-well polystyrene plate. The test compounds were first serially diluted in DMSO and the ...More data for this Ligand-Target Pair