BDBM577148 8-Cyclopropyl-10-(6-methoxypyridin-3-yl)-7,8-dihydropyrido[2',3':4,5]pyrrolo[1,2-a]pyrazin-9(6H)-one::US11472805, Example 53

SMILES COc1ccc(cn1)-c1c2C(=O)N(CCn2c2cccnc12)C1CC1

InChI Key InChIKey=FPIUDCHSBHCGEP-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 577148   

LigandPNGBDBM577148(8-Cyclopropyl-10-(6-methoxypyridin-3-yl)-7,8-dihyd...)
Affinity DataIC50:  426nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B [122-736](Homo sapiens (Human))
Pfizer

US Patent
LigandPNGBDBM577148(8-Cyclopropyl-10-(6-methoxypyridin-3-yl)-7,8-dihyd...)
Affinity DataIC50:  6.54nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent