BDBM60536 BDBM50399283::US9102622, 13.2
SMILES FS(=O)(=O)CCCCCCCc1cccc(OCc2ccccc2)c1
InChI Key InChIKey=CEOCDYLHZFETSF-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 60536
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University of Connecticut
US Patent
University of Connecticut
US Patent
Affinity DataKi: 39nM ΔG°: -10.5kcal/mole IC50: 165nMT: 2°CAssay Description:All compound solutions are made to a concentration of 10 mM in DMSO. To test the stability of the compounds in enzyme assay conditions, 25 nmoles of ...More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University of Connecticut
US Patent
University of Connecticut
US Patent
Affinity DataKi: 39nM ΔG°: -10.5kcal/mole IC50: 165nMT: 2°CAssay Description:All compound solutions are made to a concentration of 10 mM in DMSO. To test the stability of the compounds in enzyme assay conditions, 25 nmoles of ...More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University of Connecticut
US Patent
University of Connecticut
US Patent
Affinity DataKi: 46nM ΔG°: -10.4kcal/mole IC50: 193nMT: 2°CAssay Description:All compound solutions are made to a concentration of 10 mM in DMSO. To test the stability of the compounds in enzyme assay conditions, 25 nmoles of ...More data for this Ligand-Target Pair
Affinity DataKi: 99nMAssay Description:Displacement of [3H]CP-55,940 from mouse CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 335nMAssay Description:Displacement of [3H]CP-55,940 from CB1 receptor in rat brain homogenatesMore data for this Ligand-Target Pair
Affinity DataIC50: 752nMAssay Description:Inhibition of recombinant human hexahistidine-tagged MGL expressed in Escherichia coli using AHMMCE as substrate after 15 mins by medium throughput f...More data for this Ligand-Target Pair