BDBM615294 US20230271949, Example 85

SMILES Fc1cc(Cl)ccc1COc1cccc(n1)C1CCN(Cc2nc3cc(NC(=O)c4ccc5[nH]c(=O)[nH]c5c4)ccc3n2C[C@@H]2CCO2)CC1

InChI Key InChIKey=DRBYATWEGOQFAP-MHZLTWQESA-N

Data  1 KI  1 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 615294   

TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Ascletis Bioscience

US Patent
LigandPNGBDBM615294(US20230271949, Example 85)
Affinity DataKi:  71.7nMAssay Description:Tag-Lite Binding Assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Ascletis Bioscience

US Patent
LigandPNGBDBM615294(US20230271949, Example 85)
Affinity DataEC50:  0.410nMAssay Description:cAMP Detection Kit, Cisbio (Cat #62AM4PEJ).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Ascletis Bioscience

US Patent
LigandPNGBDBM615294(US20230271949, Example 85)
Affinity DataIC50:  143nMAssay Description:Tag-Lite Binding Assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent