BDBM92403 PDK1 inhibitor, 4
SMILES COc1ccc(cc1)C#Cc1ccc2ncc3ncn(-c4ccc(CCN)cc4)c3c2c1
InChI Key InChIKey=YKDDVFSLJZJKFP-UHFFFAOYSA-N
Data 1 EC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 92403
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Merck Research Laboratories
Merck Research Laboratories
Affinity DataEC50: 200nMAssay Description:Enzyme potency (PDK1 EC50)was determined using recombinant, purified full-length human PDK1 enzyme and AKT-Thr-308-tide as substrate.More data for this Ligand-Target Pair