Compile Data Set for Download or QSAR
Report error Found 523 Enz. Inhib. hit(s) with Target = '3-oxoacyl-[acyl-carrier-protein] synthase 3'
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245828BDBM50245828(2-Tosylnaphthalene-1,4-diol | CHEMBL509952)
Affinity DataIC50: 0.610nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245923BDBM50245923(2-(naphthalen-2-ylsulfonyl)naphthalene-1,4-diol | ...)
Affinity DataIC50: 1.49nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245928BDBM50245928(2-tosylnaphthalene-1,4-dione | CHEMBL454282)
Affinity DataIC50: 1.99nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245877BDBM50245877(2-(phenylsulfonyl)naphthalene-1,4-diol | CHEMBL462...)
Affinity DataIC50: 2.84nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Streptococcus pyogenes serotype M3)
Quorex Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 23585BDBM23585(2-{[4-(4-methanesulfonylphenyl)-3-phenoxybenzene]a...)
Affinity DataIC50: 3nMpH: 7.0 T: 2°CAssay Description:The potency of FabH inhibition (IC50) was determined using [3H]- or [14C]-radiolabeled substrates. This was accomplished at fixed concentrations of a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245880BDBM50245880(2-(4-propylphenylsulfonyl)naphthalene-1,4-diol | C...)
Affinity DataIC50: 3.09nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245829BDBM50245829(2-(methylsulfonyl)naphthalene-1,4-diol | CHEMBL491...)
Affinity DataIC50: 3.53nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245830BDBM50245830(3-(1,4-dihydroxynaphthalen-2-ylsulfonyl)propanoic ...)
Affinity DataIC50: 3.53nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245879BDBM50245879(2-(4-chlorophenylsulfonyl)naphthalene-1,4-diol | C...)
Affinity DataIC50: 3.61nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245878BDBM50245878(N-(4-(1,4-dihydroxynaphthalen-2-ylsulfonyl)phenyl)...)
Affinity DataIC50: 3.76nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 23587BDBM23587(2-hydroxy-6-[(3-phenoxy-4-phenylbenzene)amido]benz...)
Affinity DataIC50: 4nMpH: 7.0 T: 2°CAssay Description:The potency of FabH inhibition (IC50) was determined using [3H]- or [14C]-radiolabeled substrates. This was accomplished at fixed concentrations of a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Streptococcus pyogenes serotype M3)
Quorex Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 23587BDBM23587(2-hydroxy-6-[(3-phenoxy-4-phenylbenzene)amido]benz...)
Affinity DataIC50: 4nMpH: 7.0 T: 2°CAssay Description:The potency of FabH inhibition (IC50) was determined using [3H]- or [14C]-radiolabeled substrates. This was accomplished at fixed concentrations of a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 50412347BDBM50412347(CHEMBL499343)
Affinity DataIC50: 4nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245924BDBM50245924(2-tosylanthracene-1,4-diol | CHEMBL451059)
Affinity DataIC50: 8.47nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Escherichia coli)
Konkuk University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50276580BDBM50276580(4-((cyclohexylimino)methyl)benzene-1,3-diol | CHEM...)
Affinity DataKd:  20nMAssay Description:Binding affinity to Escherichia coli K12 KAS 3 expressed in Escherichia coli BL21 by fluorescence quenching analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 23585BDBM23585(2-{[4-(4-methanesulfonylphenyl)-3-phenoxybenzene]a...)
Affinity DataIC50: 28nMpH: 7.0 T: 2°CAssay Description:The potency of FabH inhibition (IC50) was determined using [3H]- or [14C]-radiolabeled substrates. This was accomplished at fixed concentrations of a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 23585BDBM23585(2-{[4-(4-methanesulfonylphenyl)-3-phenoxybenzene]a...)
Affinity DataIC50: 28.1nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245926BDBM50245926(cid_257482 | CHEMBL462376 | N-(4-(2,5-dihydroxyphe...)
Affinity DataIC50: 31.4nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Streptococcus pyogenes serotype M3)
Quorex Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 23586BDBM23586(2-[(4-bromo-3-phenoxybenzene)amido]-6-hydroxybenzo...)
Affinity DataIC50: 34nMpH: 7.0 T: 2°CAssay Description:The potency of FabH inhibition (IC50) was determined using [3H]- or [14C]-radiolabeled substrates. This was accomplished at fixed concentrations of a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245925BDBM50245925(2-tosylbenzene-1,4-diol | CHEMBL462375)
Affinity DataIC50: 34.4nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Streptococcus pyogenes serotype M3)
Quorex Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 23584BDBM23584(2-[(3-phenoxy-4-phenylbenzene)amido]benzoic acid |...)
Affinity DataIC50: 50nMpH: 7.0 T: 2°CAssay Description:The potency of FabH inhibition (IC50) was determined using [3H]- or [14C]-radiolabeled substrates. This was accomplished at fixed concentrations of a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 23584BDBM23584(2-[(3-phenoxy-4-phenylbenzene)amido]benzoic acid |...)
Affinity DataIC50: 56.0nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 23584BDBM23584(2-[(3-phenoxy-4-phenylbenzene)amido]benzoic acid |...)
Affinity DataIC50: 56nMpH: 7.0 T: 2°CAssay Description:The potency of FabH inhibition (IC50) was determined using [3H]- or [14C]-radiolabeled substrates. This was accomplished at fixed concentrations of a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 23586BDBM23586(2-[(4-bromo-3-phenoxybenzene)amido]-6-hydroxybenzo...)
Affinity DataIC50: 62nMpH: 7.0 T: 2°CAssay Description:The potency of FabH inhibition (IC50) was determined using [3H]- or [14C]-radiolabeled substrates. This was accomplished at fixed concentrations of a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 50412351BDBM50412351(CHEMBL499342)
Affinity DataIC50: 62.1nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 23595BDBM23595(2-({3-phenoxy-4-[4-(trifluoromethyl)phenyl]benzene...)
Affinity DataIC50: 95.9nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 23595BDBM23595(2-({3-phenoxy-4-[4-(trifluoromethyl)phenyl]benzene...)
Affinity DataIC50: 96nMAssay Description:The potency of FabH inhibition (IC50) was determined using [3H]- or [14C]-radiolabeled substrates. This was accomplished at fixed concentrations of a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 23594BDBM23594(2-{[3-phenoxy-4-(pyridin-3-yl)benzene]amido}benzoi...)
Affinity DataIC50: 110nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 23594BDBM23594(2-{[3-phenoxy-4-(pyridin-3-yl)benzene]amido}benzoi...)
Affinity DataIC50: 110nMAssay Description:The potency of FabH inhibition (IC50) was determined using [3H]- or [14C]-radiolabeled substrates. This was accomplished at fixed concentrations of a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245831BDBM50245831(2-(p-tolylthio)naphthalene-1,4-dione | CHEMBL50155...)
Affinity DataIC50: 112nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Portland State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245927BDBM50245927(2-tosylnaphthalene | CHEMBL462553)
Affinity DataIC50: 138nMAssay Description:Inhibition of Mycobacterium tuberculosis FabHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 23606BDBM23606(2-{[4-(2,4-difluorophenyl)-3-phenoxybenzene]amido}...)
Affinity DataIC50: 160nMAssay Description:The potency of FabH inhibition (IC50) was determined using [3H]- or [14C]-radiolabeled substrates. This was accomplished at fixed concentrations of a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 23596BDBM23596(2-{[4-(4-methylphenyl)-3-phenoxybenzene]amido}benz...)
Affinity DataIC50: 160nMAssay Description:The potency of FabH inhibition (IC50) was determined using [3H]- or [14C]-radiolabeled substrates. This was accomplished at fixed concentrations of a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 23596BDBM23596(2-{[4-(4-methylphenyl)-3-phenoxybenzene]amido}benz...)
Affinity DataIC50: 160nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 23606BDBM23606(2-{[4-(2,4-difluorophenyl)-3-phenoxybenzene]amido}...)
Affinity DataIC50: 160nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 23599BDBM23599(2-{[4-(4-ethoxyphenyl)-3-phenoxybenzene]amido}benz...)
Affinity DataIC50: 220nMAssay Description:The potency of FabH inhibition (IC50) was determined using [3H]- or [14C]-radiolabeled substrates. This was accomplished at fixed concentrations of a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 23599BDBM23599(2-{[4-(4-ethoxyphenyl)-3-phenoxybenzene]amido}benz...)
Affinity DataIC50: 220nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 23602BDBM23602(2-{[4-(4-fluoro-3-methylphenyl)-3-phenoxybenzene]a...)
Affinity DataIC50: 240nMAssay Description:The potency of FabH inhibition (IC50) was determined using [3H]- or [14C]-radiolabeled substrates. This was accomplished at fixed concentrations of a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 23602BDBM23602(2-{[4-(4-fluoro-3-methylphenyl)-3-phenoxybenzene]a...)
Affinity DataIC50: 240nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 23605BDBM23605(2-{[4-(4-chloro-3-methylphenyl)-3-phenoxybenzene]a...)
Affinity DataIC50: 250nMAssay Description:The potency of FabH inhibition (IC50) was determined using [3H]- or [14C]-radiolabeled substrates. This was accomplished at fixed concentrations of a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 23605BDBM23605(2-{[4-(4-chloro-3-methylphenyl)-3-phenoxybenzene]a...)
Affinity DataIC50: 250nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 23592BDBM23592(2-{[4-(3,5-dimethylpiperidin-1-yl)-3-phenoxybenzen...)
Affinity DataIC50: 270nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 23592BDBM23592(2-{[4-(3,5-dimethylpiperidin-1-yl)-3-phenoxybenzen...)
Affinity DataIC50: 270nMAssay Description:The potency of FabH inhibition (IC50) was determined using [3H]- or [14C]-radiolabeled substrates. This was accomplished at fixed concentrations of a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 23591BDBM23591(2-{[3-phenoxy-4-(piperidin-1-yl)benzene]amido}benz...)
Affinity DataIC50: 290nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 23591BDBM23591(2-{[3-phenoxy-4-(piperidin-1-yl)benzene]amido}benz...)
Affinity DataIC50: 290nMAssay Description:The potency of FabH inhibition (IC50) was determined using [3H]- or [14C]-radiolabeled substrates. This was accomplished at fixed concentrations of a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 23604BDBM23604(2-{[4-(3,4-difluorophenyl)-3-phenoxybenzene]amido}...)
Affinity DataIC50: 330nMAssay Description:The potency of FabH inhibition (IC50) was determined using [3H]- or [14C]-radiolabeled substrates. This was accomplished at fixed concentrations of a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 23604BDBM23604(2-{[4-(3,4-difluorophenyl)-3-phenoxybenzene]amido}...)
Affinity DataIC50: 330nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 23612BDBM23612(2-hydroxy-6-[(3-phenoxybenzene)amido]benzoic acid ...)
Affinity DataIC50: 410nMAssay Description:The potency of FabH inhibition (IC50) was determined using [3H]- or [14C]-radiolabeled substrates. This was accomplished at fixed concentrations of a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 23598BDBM23598(2-{[4-(4-hydroxyphenyl)-3-phenoxybenzene]amido}ben...)
Affinity DataIC50: 410nMAssay Description:The potency of FabH inhibition (IC50) was determined using [3H]- or [14C]-radiolabeled substrates. This was accomplished at fixed concentrations of a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2008
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 3(Enterococcus faecalis (strain ATCC 700802 / V583))
Quorex Pharmaceuticals

LigandChemical structure of BindingDB Monomer ID 23598BDBM23598(2-{[4-(4-hydroxyphenyl)-3-phenoxybenzene]amido}ben...)
Affinity DataIC50: 410nMAssay Description:Inhibition of Enterococcus faecalis FabH by FabD/FabH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
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