Compile Data Set for Download or QSAR
Report error Found 922 Enz. Inhib. hit(s) with Target = 'Bombesin receptor subtype-3'
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127518(peptidomimetic | CHEMBL57104)
Affinity DataEC50:  0.190nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50275902(D-Phe-Gln-Trp-Ala-Val-b-Ala-His-Phe-Nle-NH2 | CHEM...)
Affinity DataKi:  0.360nMAssay Description:Binding affinity to BRS-3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50381918(CHEMBL2023113)
Affinity DataIC50: 0.5nMAssay Description:Displacement of 125I-dY-peptide from human BRS3 expressed in NFAT-CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50381917(CHEMBL2023112)
Affinity DataIC50: 0.5nMAssay Description:Displacement of 125I-dY-peptide from human BRS3 expressed in NFAT-CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50336889((2S)-1,1,1-trifluoro-2-[4-(1H-pyrazol-1-yl)phenyl]...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]Bag-3 from rat BRS-3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50336889((2S)-1,1,1-trifluoro-2-[4-(1H-pyrazol-1-yl)phenyl]...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]Bag-3 from rat BRS-3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50381916(CHEMBL2023111)
Affinity DataIC50: 0.600nMAssay Description:Displacement of 125I-dY-peptide from human BRS3 expressed in NFAT-CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50400247(CHEMBL2179918)
Affinity DataIC50: 0.700nMAssay Description:Displacement of [125I]-[D-Tyr6,beta-Ala11,Phe13,Nle14]-Bombesin(6-14) from human BRS3 expressed in CHO cells expressing NFAT after 2 hrs by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50394612(CHEMBL2164581)
Affinity DataIC50: 0.700nMAssay Description:Displacement of [125I]-dY-peptide from human BRS-3 expressed in NFAT-CHO cells after 2 hrs by by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50394616(CHEMBL2164577)
Affinity DataIC50: 0.760nMAssay Description:Displacement of [125I]-dY-peptide from human BRS-3 expressed in NFAT-CHO cells after 2 hrs by by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50533323(CHEMBL4435571)
Affinity DataEC50:  0.800nMAssay Description:Agonist activity at mouse BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50533323(CHEMBL4435571)
Affinity DataEC50:  0.800nMAssay Description:Agonist activity at mouse BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM86502(NSC_0 | CAS_0 | [D-Tyr6,Beta-Ala11,Phe13,Nle14]Bn(...)
Affinity DataKi:  0.820nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2012
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50533323(CHEMBL4435571)
Affinity DataEC50:  0.900nMAssay Description:Agonist activity at human BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50533323(CHEMBL4435571)
Affinity DataEC50:  0.900nMAssay Description:Agonist activity at human BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50394609(CHEMBL2164223)
Affinity DataIC50: 0.900nMAssay Description:Displacement of [125I]-dY-peptide from human BRS-3 expressed in NFAT-CHO cells after 2 hrs by by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50400254(CHEMBL2179911)
Affinity DataIC50: 0.900nMAssay Description:Displacement of [125I]-[D-Tyr6,beta-Ala11,Phe13,Nle14]-Bombesin(6-14) from human BRS3 expressed in CHO cells expressing NFAT after 2 hrs by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50533327(CHEMBL4461212)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50447496(CHEMBL3115400)
Affinity DataEC50:  1nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50447496(CHEMBL3115400)
Affinity DataEC50:  1nMAssay Description:Agonist activity at mouse BRS-3 expressed in CHOK1 cells after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50533327(CHEMBL4461212)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50158702(Universal ligand | CHEMBL413893)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of bombesin subtype 3 receptor expressed in human lung carcinoidsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50394613(CHEMBL2164580)
Affinity DataIC50: 1.10nMAssay Description:Displacement of [125I]-dY-peptide from human BRS-3 expressed in NFAT-CHO cells after 2 hrs by by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50394611(CHEMBL2164582)
Affinity DataIC50: 1.20nMAssay Description:Displacement of [125I]-dY-peptide from human BRS-3 expressed in NFAT-CHO cells after 2 hrs by by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50400257(CHEMBL2179908)
Affinity DataIC50: 1.20nMAssay Description:Displacement of [125I]-[D-Tyr6,beta-Ala11,Phe13,Nle14]-Bombesin(6-14) from human BRS3 expressed in CHO cells expressing NFAT after 2 hrs by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50447496(CHEMBL3115400)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at human BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50447496(CHEMBL3115400)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at human BRS-3 expressed in CHOK1 cells after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50381914(MK-7725 | CHEMBL2023109)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at human BRS-3 expressed in CHOK1 cells after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127544(peptidomimetic | CHEMBL56369)
Affinity DataEC50:  1.40nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50394615(CHEMBL2164578)
Affinity DataIC50: 1.40nMAssay Description:Displacement of [125I]-dY-peptide from human BRS-3 expressed in NFAT-CHO cells after 2 hrs by by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50381915(CHEMBL2023110)
Affinity DataIC50: 1.40nMAssay Description:Displacement of 125I-dY-peptide from human BRS3 expressed in NFAT-CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127520(peptidomimetic | CHEMBL57438)
Affinity DataEC50:  1.5nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50447479(CHEMBL3115386)
Affinity DataEC50:  1.60nMAssay Description:Agonist activity at human BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50400246(CHEMBL2179473)
Affinity DataIC50: 1.60nMAssay Description:Displacement of [125I]-[D-Tyr6,beta-Ala11,Phe13,Nle14]-Bombesin(6-14) from human BRS3 expressed in CHO cells expressing NFAT after 2 hrs by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50336889((2S)-1,1,1-trifluoro-2-[4-(1H-pyrazol-1-yl)phenyl]...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]Bag-3 from mouse BRS-3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50447479(CHEMBL3115386)
Affinity DataEC50:  1.60nMAssay Description:Agonist activity at human BRS-3 expressed in CHOK1 cells after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50447475(CHEMBL3115390)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at human BRS-3 expressed in CHOK1 cells after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50447475(CHEMBL3115390)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at human BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50394608(CHEMBL2164224)
Affinity DataIC50: 1.70nMAssay Description:Displacement of [125I]-dY-peptide from human BRS-3 expressed in NFAT-CHO cells after 2 hrs by by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50447477(CHEMBL3115388)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at human BRS-3 expressed in CHOK1 cells after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50447477(CHEMBL3115388)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at human BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2016
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50394617(CHEMBL2164576)
Affinity DataIC50: 1.72nMAssay Description:Displacement of [125I]-dY-peptide from human BRS-3 expressed in NFAT-CHO cells after 2 hrs by by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50394610(CHEMBL2164222)
Affinity DataIC50: 1.90nMAssay Description:Displacement of [125I]-dY-peptide from human BRS-3 expressed in NFAT-CHO cells after 2 hrs by by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50533320(CHEMBL4580739)
Affinity DataEC50:  2nMAssay Description:Agonist activity at mouse BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50533331(CHEMBL4448589)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50533320(CHEMBL4580739)
Affinity DataEC50:  2nMAssay Description:Agonist activity at mouse BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50533331(CHEMBL4448589)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50381919(CHEMBL2023114)
Affinity DataIC50: 2.10nMAssay Description:Displacement of 125I-dY-peptide from human BRS3 expressed in NFAT-CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127539(3-(1H-Indol-3-yl)-N-phenethyl-2-(2-phenylacetylami...)
Affinity DataEC50:  2.10nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127527(peptidomimetic | CHEMBL294647)
Affinity DataEC50:  2.20nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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