Compile Data Set for Download or QSAR
Report error Found 90 Enz. Inhib. hit(s) with Target = 'Calmodulin-1'
TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 59172BDBM59172(BN2)
Affinity DataKd:  10nMAssay Description:Experiments were conducted with HITACHI-4500 and Shimadzu RF-5301 fluorescence spectrophotometer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2011
Entry Details Article
PubMed
TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 50260600BDBM50260600(N-(3,3,-DIPHENYLPROPYL)-N'-[1-R-(2 3,4-BIS-BUTOXYP...)
Affinity DataKd:  18nMAssay Description:Binding affinity to calmodulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 59171BDBM59171(BN1)
Affinity DataKd:  70nMAssay Description:Experiments were conducted with HITACHI-4500 and Shimadzu RF-5301 fluorescence spectrophotometer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2011
Entry Details Article
PubMed
TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 50652792BDBM50652792(CHEMBL3752910)
Affinity DataKd:  110nMAssay Description:Binding affinity to human CALM1 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 50652793BDBM50652793(CHEMBL5653589)
Affinity DataKd:  213nMAssay Description:Binding affinity to human CALM1 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 588519BDBM588519(US11542290, Compound MT-035)
Affinity DataIC50: 240nMAssay Description:The competition binding assay was performed in a 384-well plate format and in 20 μl reactions. Serial dilutions (0.001-100 μM) of a test co...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 588481BDBM588481(US11542290, Compound A-7)
Affinity DataIC50: 470nMAssay Description:The competition binding assay was performed in a 384-well plate format and in 20 μl reactions. Serial dilutions (0.001-100 μM) of a test co...More data for this Ligand-Target Pair
Ligand InfoPurchaseSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 588520BDBM588520(US11542290, Compound MT-037 | US11542290, Compound...)
Affinity DataIC50: 850nMAssay Description:The competition binding assay was performed in a 384-well plate format and in 20 μl reactions. Serial dilutions (0.001-100 μM) of a test co...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 588491BDBM588491(US11542290, Compound MT-009)
Affinity DataIC50: 860nMAssay Description:The competition binding assay was performed in a 384-well plate format and in 20 μl reactions. Serial dilutions (0.001-100 μM) of a test co...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 588490BDBM588490(US11542290, Compound MT-008)
Affinity DataIC50: 900nMAssay Description:The competition binding assay was performed in a 384-well plate format and in 20 μl reactions. Serial dilutions (0.001-100 μM) of a test co...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 79181BDBM79181(cid_2913535 | TRIFLUOPERAZINE | SMR000059133 | MLS...)
Affinity DataKd:  1.00E+3nMAssay Description:Binding affinity to calmodulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 588513BDBM588513(US11542290, Compound MT-030a)
Affinity DataIC50: 1.01E+3nMAssay Description:The competition binding assay was performed in a 384-well plate format and in 20 μl reactions. Serial dilutions (0.001-100 μM) of a test co...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 79181BDBM79181(cid_2913535 | TRIFLUOPERAZINE | SMR000059133 | MLS...)
Affinity DataIC50: 1.06E+3nMAssay Description:The competition binding assay was performed in a 384-well plate format and in 20 μl reactions. Serial dilutions (0.001-100 μM) of a test co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 79181BDBM79181(cid_2913535 | TRIFLUOPERAZINE | SMR000059133 | MLS...)
Affinity DataIC50: 1.06E+3nMAssay Description:The competition binding assay was performed in a 384-well plate format and in 20 μl reactions. Serial dilutions (0.001-100 μM) of a test co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 79181BDBM79181(cid_2913535 | TRIFLUOPERAZINE | SMR000059133 | MLS...)
Affinity DataIC50: 1.11E+3nMAssay Description:The competition binding assay was performed in a 384-well plate format and in 20 μl reactions. Serial dilutions (0.001-100 μM) of a test co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 588484BDBM588484(US11542290, Compound MT-002)
Affinity DataIC50: 1.41E+3nMAssay Description:The competition binding assay was performed in a 384-well plate format and in 20 μl reactions. Serial dilutions (0.001-100 μM) of a test co...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 588512BDBM588512(US11542290, Compound MT-030)
Affinity DataIC50: 1.65E+3nMAssay Description:The competition binding assay was performed in a 384-well plate format and in 20 μl reactions. Serial dilutions (0.001-100 μM) of a test co...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 588485BDBM588485(US11542290, Compound MT-003)
Affinity DataIC50: 1.73E+3nMAssay Description:The competition binding assay was performed in a 384-well plate format and in 20 μl reactions. Serial dilutions (0.001-100 μM) of a test co...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 588508BDBM588508(US11542290, Compound MT-026)
Affinity DataIC50: 2.03E+3nMAssay Description:The competition binding assay was performed in a 384-well plate format and in 20 μl reactions. Serial dilutions (0.001-100 μM) of a test co...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 588501BDBM588501(US11542290, Compound MT-019)
Affinity DataIC50: 2.83E+3nMAssay Description:The competition binding assay was performed in a 384-well plate format and in 20 μl reactions. Serial dilutions (0.001-100 μM) of a test co...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 588515BDBM588515(US11542290, Compound MT-031a)
Affinity DataIC50: 2.97E+3nMAssay Description:The competition binding assay was performed in a 384-well plate format and in 20 μl reactions. Serial dilutions (0.001-100 μM) of a test co...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 588489BDBM588489(US11542290, Compound MT-007)
Affinity DataIC50: 2.97E+3nMAssay Description:The competition binding assay was performed in a 384-well plate format and in 20 μl reactions. Serial dilutions (0.001-100 μM) of a test co...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 588520BDBM588520(US11542290, Compound MT-037 | US11542290, Compound...)
Affinity DataIC50: 2.99E+3nMAssay Description:The competition binding assay was performed in a 384-well plate format and in 20 μl reactions. Serial dilutions (0.001-100 μM) of a test co...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 588487BDBM588487(US11542290, Compound MT-005)
Affinity DataIC50: 3.17E+3nMAssay Description:The competition binding assay was performed in a 384-well plate format and in 20 μl reactions. Serial dilutions (0.001-100 μM) of a test co...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 588522BDBM588522(US11542290, Compound MT-038)
Affinity DataIC50: 3.90E+3nMAssay Description:The competition binding assay was performed in a 384-well plate format and in 20 μl reactions. Serial dilutions (0.001-100 μM) of a test co...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 588505BDBM588505(US11542290, Compound MT-023)
Affinity DataIC50: 3.96E+3nMAssay Description:The competition binding assay was performed in a 384-well plate format and in 20 μl reactions. Serial dilutions (0.001-100 μM) of a test co...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 588518BDBM588518(US11542290, Compound MT-034)
Affinity DataIC50: 4.10E+3nMAssay Description:The competition binding assay was performed in a 384-well plate format and in 20 μl reactions. Serial dilutions (0.001-100 μM) of a test co...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 588493BDBM588493(US11542290, Compound MT-011)
Affinity DataIC50: 4.47E+3nMAssay Description:The competition binding assay was performed in a 384-well plate format and in 20 μl reactions. Serial dilutions (0.001-100 μM) of a test co...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 588510BDBM588510(US11542290, Compound MT-028)
Affinity DataIC50: 4.83E+3nMAssay Description:The competition binding assay was performed in a 384-well plate format and in 20 μl reactions. Serial dilutions (0.001-100 μM) of a test co...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 588517BDBM588517(US11542290, Compound MT-033)
Affinity DataIC50: 4.99E+3nMAssay Description:The competition binding assay was performed in a 384-well plate format and in 20 μl reactions. Serial dilutions (0.001-100 μM) of a test co...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 50081950BDBM50081950(6-hydroxy-2-phenyl-4H-chromen-4-one | NSC-26744 | ...)
Affinity DataIC50: 5.17E+3nMAssay Description:Inhibition of human recombinant calmodulin assessed as inhibition of calmodulin-sensitive cAMP phosphodiesterase activation after 15 mins by spectrop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 50266274BDBM50266274(14-methoxytajixanthone | CHEMBL515370)
Affinity DataIC50: 5.54E+3nMAssay Description:Inhibition of recombinant calmodulin mediated bovine brain PDE1 activation assessed as effect on inorganic phosphate release by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 50266275BDBM50266275(Tajixanthone hydrate | CHEMBL456494)
Affinity DataIC50: 5.62E+3nMAssay Description:Inhibition of recombinant calmodulin mediated bovine brain PDE1 activation assessed as effect on inorganic phosphate release by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 588494BDBM588494(US11542290, Compound MT-012)
Affinity DataIC50: 5.65E+3nMAssay Description:The competition binding assay was performed in a 384-well plate format and in 20 μl reactions. Serial dilutions (0.001-100 μM) of a test co...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 588507BDBM588507(US11542290, Compound MT-025)
Affinity DataIC50: 6.70E+3nMAssay Description:The competition binding assay was performed in a 384-well plate format and in 20 μl reactions. Serial dilutions (0.001-100 μM) of a test co...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 588506BDBM588506(US11542290, Compound MT-024)
Affinity DataIC50: 7.02E+3nMAssay Description:The competition binding assay was performed in a 384-well plate format and in 20 μl reactions. Serial dilutions (0.001-100 μM) of a test co...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 50001888BDBM50001888([3-(2-Chloro-phenothiazin-10-yl)-propyl]-dimethyl-...)
Affinity DataIC50: 7.26E+3nMAssay Description:Inhibition of recombinant calmodulin mediated bovine brain PDE1 activation assessed as effect on inorganic phosphate release by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 588516BDBM588516(US11542290, Compound MT-032)
Affinity DataIC50: 7.43E+3nMAssay Description:The competition binding assay was performed in a 384-well plate format and in 20 μl reactions. Serial dilutions (0.001-100 μM) of a test co...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 588498BDBM588498(US11542290, Compound MT-016)
Affinity DataIC50: 7.82E+3nMAssay Description:The competition binding assay was performed in a 384-well plate format and in 20 μl reactions. Serial dilutions (0.001-100 μM) of a test co...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 588503BDBM588503(US11542290, Compound MT-021)
Affinity DataIC50: 8.13E+3nMAssay Description:The competition binding assay was performed in a 384-well plate format and in 20 μl reactions. Serial dilutions (0.001-100 μM) of a test co...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 588514BDBM588514(US11542290, Compound MT-031)
Affinity DataIC50: 8.93E+3nMAssay Description:The competition binding assay was performed in a 384-well plate format and in 20 μl reactions. Serial dilutions (0.001-100 μM) of a test co...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 59170BDBM59170(BT2)
Affinity DataKd:  9.00E+3nMAssay Description:Experiments were conducted with HITACHI-4500 and Shimadzu RF-5301 fluorescence spectrophotometer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2011
Entry Details Article
PubMed
TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 588509BDBM588509(US11542290, Compound MT-027)
Affinity DataIC50: 9.03E+3nMAssay Description:The competition binding assay was performed in a 384-well plate format and in 20 μl reactions. Serial dilutions (0.001-100 μM) of a test co...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 50346822BDBM50346822(CHEMBL66917)
Affinity DataIC50: 9.38E+3nMAssay Description:Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 minMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 50266273BDBM50266273(15-chlorotajixanthone hydrate | CHEMBL458017)
Affinity DataIC50: 9.59E+3nMAssay Description:Inhibition of recombinant calmodulin mediated bovine brain PDE1 activation assessed as effect on inorganic phosphate release by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 588496BDBM588496(US11542290, Compound MT-014)
Affinity DataIC50: 9.60E+3nMAssay Description:The competition binding assay was performed in a 384-well plate format and in 20 μl reactions. Serial dilutions (0.001-100 μM) of a test co...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 59169BDBM59169(BT1)
Affinity DataKd:  1.00E+4nMAssay Description:Experiments were conducted with HITACHI-4500 and Shimadzu RF-5301 fluorescence spectrophotometer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2011
Entry Details Article
PubMed
TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 50001888BDBM50001888([3-(2-Chloro-phenothiazin-10-yl)-propyl]-dimethyl-...)
Affinity DataIC50: 1.03E+4nMAssay Description:Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 minMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 7460BDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-chromone;...)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of human recombinant calmodulin assessed as inhibition of calmodulin-sensitive cAMP phosphodiesterase activation after 15 mins by spectrop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetCalmodulin-1(Human)
University of Sheffield

LigandChemical structure of BindingDB Monomer ID 588502BDBM588502(US11542290, Compound MT-020)
Affinity DataIC50: 1.39E+4nMAssay Description:The competition binding assay was performed in a 384-well plate format and in 20 μl reactions. Serial dilutions (0.001-100 μM) of a test co...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
US Patent

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