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Report error Found 55 Enz. Inhib. hit(s) with Target = 'Cytosol aminopeptidase [33-68,L62W]'
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50025043BDBM50025043(CHEMBL3355104)
Affinity DataKi:  20nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50457473BDBM50457473(CHEMBL4209822)
Affinity DataIC50: 30nMAssay Description:Inhibition of porcine kidney leucine aminopeptidase using LGG as substrate after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50025041BDBM50025041(CHEMBL3355106)
Affinity DataKi:  39nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50025042BDBM50025042(CHEMBL3355105)
Affinity DataKi:  50nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50129684BDBM50129684(3-[(1-amino-3-phenyl-propyl)-hydroxy-phosphinoyl]-...)
Affinity DataKi:  66nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50129681BDBM50129681(3-[(1-Amino-3-phenyl-propyl)-hydroxy-phosphinoyl]-...)
Affinity DataKi:  67nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50025070BDBM50025070(CHEMBL3355110)
Affinity DataKi:  74nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50457466BDBM50457466(CHEMBL4206158)
Affinity DataIC50: 100nMAssay Description:Inhibition of porcine kidney leucine aminopeptidase using LGG as substrate after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50025099BDBM50025099(CHEMBL3355111)
Affinity DataKi:  108nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50025066BDBM50025066(CHEMBL3355109)
Affinity DataKi:  138nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50025044BDBM50025044(CHEMBL3355103)
Affinity DataKi:  157nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50025050BDBM50025050(CHEMBL3355108)
Affinity DataKi:  195nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50337147BDBM50337147((RS)-1-amino-3-cyclohexylpropylphosphonic acid | C...)
Affinity DataKi:  210nMAssay Description:Inhibition of porcine kidney leucine aminopeptidase M17 using Leu-AMC as substrate preincubated for 30 to 60 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2017
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50025047BDBM50025047(CHEMBL3355100)
Affinity DataKi:  213nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50025046BDBM50025046(CHEMBL3355101)
Affinity DataKi:  215nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024594BDBM50024594(LEUCINE PHOSPHONIC ACID | (R)-1-Ammonium-3-methyl-...)
Affinity DataKi:  230nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50025045BDBM50025045(CHEMBL3355102)
Affinity DataKi:  593nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50025049BDBM50025049(CHEMBL3355107)
Affinity DataKi:  1.03E+3nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 234297BDBM234297(Met-ψ[P(O)(OH)CH2]-Ala (5))
Affinity DataKi:  3.64E+3nM ΔG°:  -31.0kJ/molepH: 8.4 T: 2°CAssay Description:LAP was assayed in 75 mM triethanolamine hydrochloride buffer (pH = 8.4, containing 5 mM MgCl2) at 25°C. The substrate (L-leucine-p-nitroanilide) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50316049BDBM50316049(1-amino-3-phenylpropylphosphonic acid | CHEMBL1090...)
Affinity DataKi:  4.55E+3nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50025048BDBM50025048(CHEMBL3355099)
Affinity DataKi:  5.03E+3nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170875BDBM50170875(CHEMBL3805288)
Affinity DataKi:  7.02E+3nMAssay Description:Inhibition of porcine kidney leucine aminopeptidase M17 using Leu-AMC as substrate preincubated for 30 to 60 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2017
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078125BDBM50078125((1-Amino-3-phenyl-propyl)-phosphinic acid | CHEMBL...)
Affinity DataKi:  7.69E+3nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170881BDBM50170881(CHEMBL3805028)
Affinity DataKi:  1.52E+4nMAssay Description:Inhibition of porcine kidney leucine aminopeptidase M17 using Leu-AMC as substrate preincubated for 30 to 60 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2017
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170878BDBM50170878(CHEMBL3806197)
Affinity DataKi:  1.95E+4nMAssay Description:Inhibition of porcine kidney leucine aminopeptidase M17 using Leu-AMC as substrate preincubated for 30 to 60 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2017
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170897BDBM50170897(CHEMBL3805573)
Affinity DataKi:  2.08E+4nMAssay Description:Inhibition of porcine kidney leucine aminopeptidase M17 using Leu-AMC as substrate preincubated for 30 to 60 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2017
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170880BDBM50170880(CHEMBL3806187)
Affinity DataKi:  2.10E+4nMAssay Description:Inhibition of porcine kidney leucine aminopeptidase M17 using Leu-AMC as substrate preincubated for 30 to 60 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2017
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170884BDBM50170884(CHEMBL3805495)
Affinity DataKi:  2.11E+4nMAssay Description:Inhibition of porcine kidney leucine aminopeptidase M17 using Leu-AMC as substrate preincubated for 30 to 60 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2017
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 234295BDBM234295(Met-PH (2))
Affinity DataKi:  2.20E+4nM ΔG°:  -26.6kJ/molepH: 8.4 T: 2°CAssay Description:LAP was assayed in 75 mM triethanolamine hydrochloride buffer (pH = 8.4, containing 5 mM MgCl2) at 25°C. The substrate (L-leucine-p-nitroanilide) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 234294BDBM234294(Met-P (1))
Affinity DataKi:  2.26E+4nM ΔG°:  -26.5kJ/molepH: 8.4 T: 2°CAssay Description:LAP was assayed in 75 mM triethanolamine hydrochloride buffer (pH = 8.4, containing 5 mM MgCl2) at 25°C. The substrate (L-leucine-p-nitroanilide) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170883BDBM50170883(CHEMBL3805118)
Affinity DataKi:  2.38E+4nMAssay Description:Inhibition of porcine kidney leucine aminopeptidase M17 using Leu-AMC as substrate preincubated for 30 to 60 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2017
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170876BDBM50170876(CHEMBL3805817)
Affinity DataKi:  2.62E+4nMAssay Description:Inhibition of porcine kidney leucine aminopeptidase M17 using Leu-AMC as substrate preincubated for 30 to 60 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2017
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170877BDBM50170877(CHEMBL3804956)
Affinity DataKi:  2.65E+4nMAssay Description:Inhibition of porcine kidney leucine aminopeptidase M17 using Leu-AMC as substrate preincubated for 30 to 60 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2017
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170882BDBM50170882(CHEMBL3804856)
Affinity DataKi:  2.83E+4nMAssay Description:Inhibition of porcine kidney leucine aminopeptidase M17 using Leu-AMC as substrate preincubated for 30 to 60 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2017
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 7460BDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-chromone;...)
Affinity DataIC50: 3.43E+4nMAssay Description:Inhibition of pig kidney cytosolic Leucyl aminopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157555BDBM50157555(2-(3,4-dihydroxyphenyl)-4H-chromen-4-one | 3',4'-d...)
Affinity DataIC50: 3.51E+4nMAssay Description:Inhibition of pig kidney cytosolic Leucyl aminopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 7459BDBM7459(2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4H-chromen-4...)
Affinity DataIC50: 4.96E+4nMAssay Description:Inhibition of pig kidney cytosolic Leucyl aminopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170871BDBM50170871(CHEMBL3806230)
Affinity DataKi:  5.58E+4nMAssay Description:Inhibition of porcine kidney leucine aminopeptidase M17 using Leu-AMC as substrate preincubated for 30 to 60 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2017
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50316030BDBM50316030(1-aminopentylphosphonic acid | CHEMBL1089899 | Nle...)
Affinity DataKi:  5.80E+4nM ΔG°:  -24.2kJ/molepH: 8.4 T: 2°CAssay Description:LAP was assayed in 75 mM triethanolamine hydrochloride buffer (pH = 8.4, containing 5 mM MgCl2) at 25°C. The substrate (L-leucine-p-nitroanilide) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170879BDBM50170879(CHEMBL3805472)
Affinity DataKi:  6.44E+4nMAssay Description:Inhibition of porcine kidney leucine aminopeptidase M17 using Leu-AMC as substrate preincubated for 30 to 60 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2017
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170894BDBM50170894(CHEMBL3805338)
Affinity DataKi:  6.84E+4nMAssay Description:Inhibition of porcine kidney leucine aminopeptidase M17 using Leu-AMC as substrate preincubated for 30 to 60 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2017
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170895BDBM50170895(CHEMBL3805487)
Affinity DataKi:  6.91E+4nMAssay Description:Inhibition of porcine kidney leucine aminopeptidase M17 using Leu-AMC as substrate preincubated for 30 to 60 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2017
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170873BDBM50170873(CHEMBL3805193)
Affinity DataKi:  7.11E+4nMAssay Description:Inhibition of porcine kidney leucine aminopeptidase M17 using Leu-AMC as substrate preincubated for 30 to 60 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2017
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170898BDBM50170898(CHEMBL3805964)
Affinity DataKi:  7.26E+4nMAssay Description:Inhibition of porcine kidney leucine aminopeptidase M17 using Leu-AMC as substrate preincubated for 30 to 60 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2017
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 234296BDBM234296(Nle-PH (4))
Affinity DataKi:  7.39E+4nM ΔG°:  -23.6kJ/molepH: 8.4 T: 2°CAssay Description:LAP was assayed in 75 mM triethanolamine hydrochloride buffer (pH = 8.4, containing 5 mM MgCl2) at 25°C. The substrate (L-leucine-p-nitroanilide) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170874BDBM50170874(CHEMBL3805544)
Affinity DataKi:  1.08E+5nMAssay Description:Inhibition of porcine kidney leucine aminopeptidase M17 using Leu-AMC as substrate preincubated for 30 to 60 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2017
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170900BDBM50170900(CHEMBL3806247)
Affinity DataKi:  1.19E+5nMAssay Description:Inhibition of porcine kidney leucine aminopeptidase M17 using Leu-AMC as substrate preincubated for 30 to 60 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2017
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 234299BDBM234299(Nle-ψ[P(O)(OH)O]-L-AlaOMe (7))
Affinity DataKi:  2.19E+5nM ΔG°:  -20.9kJ/molepH: 8.4 T: 2°CAssay Description:LAP was assayed in 75 mM triethanolamine hydrochloride buffer (pH = 8.4, containing 5 mM MgCl2) at 25°C. The substrate (L-leucine-p-nitroanilide) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024597BDBM50024597((S)-1-Ammonium-3-methyl-butane-1-phosphonic acid a...)
Affinity DataKi:  2.20E+5nMAssay Description:Inhibition of pig recombinant leucine aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetCytosol aminopeptidase [33-68,L62W](Pig)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50170896BDBM50170896(CHEMBL3805251)
Affinity DataKi:  2.40E+5nMAssay Description:Inhibition of porcine kidney leucine aminopeptidase M17 using Leu-AMC as substrate preincubated for 30 to 60 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2017
Entry Details Article
PubMed
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