Compile Data Set for Download or QSAR
Report error Found 307 Enz. Inhib. hit(s) with Target = 'Ecdysone receptor'
TargetEcdysone receptor/Protein ultraspiracle homolog(Spruce budworm moth)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandPNGBDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataKi:  0.501nMAssay Description:Binding affinity to Choristoneura fumiferana EcRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488460(CHEBI:38450 | Chromafenozide)
Affinity DataEC50:  1nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataEC50:  1.20nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Fruit fly)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50326776(2,3,14,20,22-PENTAHYDROXYCHOLEST-7-EN-6-ONE | Pona...)
Affinity DataIC50: 1.29nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetEcdysone receptor/Ultraspiracle(Asiatic rice borer moth)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandPNGBDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataKi:  1.30nMAssay Description:Binding affinity to Chilo suppressalis (rice stem borer) EcRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Egyptian cotton leafworm)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataEC50:  2.20nMAssay Description:Agonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Egyptian cotton leafworm)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488460(CHEBI:38450 | Chromafenozide)
Affinity DataEC50:  2.60nMAssay Description:Agonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488450(CHEMBL2286445)
Affinity DataEC50:  2.90nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor/Gene regulation protein(Tobacco budworm moth)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandPNGBDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataKi:  3.20nMAssay Description:Binding affinity to Heliothis virescens (tobacco budworm) EcRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor/USP(Indianmeal moth)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandPNGBDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataKi:  3.20nMAssay Description:Binding affinity to Plodia interpunctella (Indian meal moth ) EcRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50128305(N'-tert-butyl-N'-(3,5-dimethylbenzoyl)-3-methoxy-2...)
Affinity DataEC50:  3.40nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Egyptian cotton leafworm)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488468(CHEMBL2286448)
Affinity DataEC50:  3.40nMAssay Description:Agonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488468(CHEMBL2286448)
Affinity DataEC50:  4.40nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488468(CHEMBL2286448)
Affinity DataEC50:  4.40nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488456(CHEMBL2286431)
Affinity DataEC50:  4.90nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Egyptian cotton leafworm)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488450(CHEMBL2286445)
Affinity DataEC50:  5.40nMAssay Description:Agonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488514(CHEMBL2286720)
Affinity DataEC50:  5.80nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50128305(N'-tert-butyl-N'-(3,5-dimethylbenzoyl)-3-methoxy-2...)
Affinity DataEC50:  6nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Egyptian cotton leafworm)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50128305(N'-tert-butyl-N'-(3,5-dimethylbenzoyl)-3-methoxy-2...)
Affinity DataEC50:  6nMAssay Description:Agonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488441(CHEMBL2286428)
Affinity DataEC50:  6.60nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Egyptian cotton leafworm)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488457(CHEMBL2286430)
Affinity DataEC50:  7.10nMAssay Description:Agonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488457(CHEMBL2286430)
Affinity DataEC50:  7.10nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488508(CHEMBL2286946)
Affinity DataEC50:  7.60nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488458(CHEMBL2286427)
Affinity DataEC50:  9.10nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488482(CHEMBL2286721)
Affinity DataEC50:  9.30nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor/Ultraspiracle(Midge)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandPNGBDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataKi:  10nMAssay Description:Binding affinity to Chironomus tentans EcRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488440(CHEMBL2228849)
Affinity DataEC50:  11nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488528(CHEMBL2286728)
Affinity DataEC50:  12nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488495(CHEMBL2286703)
Affinity DataEC50:  13nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488507(CHEMBL2286723)
Affinity DataEC50:  15nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Egyptian cotton leafworm)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488440(CHEMBL2228849)
Affinity DataEC50:  16nMAssay Description:Agonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488456(CHEMBL2286431)
Affinity DataEC50:  17nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Egyptian cotton leafworm)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488441(CHEMBL2286428)
Affinity DataEC50:  17nMAssay Description:Agonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488481(CHEMBL2228859)
Affinity DataEC50:  19nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488497(CHEMBL2286719)
Affinity DataEC50:  19nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488496(CHEMBL2286722)
Affinity DataEC50:  20nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488441(CHEMBL2286428)
Affinity DataEC50:  25nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488458(CHEMBL2286427)
Affinity DataEC50:  31nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488470(CHEMBL2286444)
Affinity DataEC50:  33nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488473(CHEMBL2286426)
Affinity DataEC50:  34nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Fruit fly)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50326777((2beta,3beta,5beta,22R)-2,3,14,20,22,25-hexahydrox...)
Affinity DataIC50: 45.7nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488476(CHEMBL2286429)
Affinity DataEC50:  51nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488475(CHEMBL2286422)
Affinity DataEC50:  51nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488490(CHEMBL2286729)
Affinity DataEC50:  52nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488532(CHEMBL2286750)
Affinity DataEC50:  52nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Fruit fly)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414658(CHEMBL559048)
Affinity DataIC50: 58.9nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetEcdysone receptor(Fruit fly)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50414645(CYASTERONE)
Affinity DataIC50: 61.7nMAssay Description:Binding affinity to ecdysone receptor ligand binding domain in Drosophila melanogaster assessed as number of hydrogen bonds formedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50178985(CHEMBL2286727)
Affinity DataEC50:  66nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Egyptian cotton leafworm)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488470(CHEMBL2286444)
Affinity DataEC50:  68nMAssay Description:Agonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
Displayed 1 to 50 (of 307 total ) | Next | Last >>
Jump to: