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Found 10 Enz. Inhib. hit(s) with Target = 'Ecdysone receptor/Ultraspiracle'
TargetEcdysone receptor/Ultraspiracle(Chilo suppressalis)
Csiro Materials Science And Engineering And Csiro Food And Nutritional Sciences

Curated by ChEMBL
LigandPNGBDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataKi:  1.30nMAssay Description:Binding affinity to Chilo suppressalis (rice stem borer) EcRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor/Ultraspiracle(Chironomus tentans)
Csiro Materials Science And Engineering And Csiro Food And Nutritional Sciences

Curated by ChEMBL
LigandPNGBDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataKi:  10nMAssay Description:Binding affinity to Chironomus tentans EcRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor/Ultraspiracle protein(Lucilia cuprina)
Csiro Materials Science And Engineering And Csiro Food And Nutritional Sciences

Curated by ChEMBL
LigandPNGBDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataKi:  158nMAssay Description:Binding affinity to Lucilia cuprina EcRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor/Ultraspiracle(Anthonomus grandis)
Csiro Materials Science And Engineering And Csiro Food And Nutritional Sciences

Curated by ChEMBL
LigandPNGBDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataKi:  1.26E+4nMAssay Description:Binding affinity to Anthonomus grandis ecdysone receptor (EcR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor/Ultraspiracle protein(Myzus persicae)
Csiro Materials Science And Engineering And Csiro Food And Nutritional Sciences

Curated by ChEMBL
LigandPNGBDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataKi: <1.26E+5nMAssay Description:Binding affinity to Myzus persicae EcR (green peach aphid)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor/Ultraspiracle protein(Bemisia tabaci)
Csiro Materials Science And Engineering And Csiro Food And Nutritional Sciences

Curated by ChEMBL
LigandPNGBDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataKi: <5.01E+5nMAssay Description:Binding affinity to Bemisia tabaci (sweet potato whitefly) ecdysone receptor (EcR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor/Ultraspiracle protein(Spodoptera frugiperda)
Csiro Materials Science And Engineering And Csiro Food And Nutritional Sciences

Curated by ChEMBL
LigandPNGBDBM50226672(CHEMBL255034 | makisterone A)
Affinity DataIC50:  389nMAssay Description:Binding affinity to Spodoptera frugiperda (fall armyworm) EcRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor/Ultraspiracle(Leptinotarsa decemlineata)
Csiro Materials Science And Engineering And Csiro Food And Nutritional Sciences

Curated by ChEMBL
LigandPNGBDBM50326777((2beta,3beta,5beta,22R)-2,3,14,20,22,25-hexahydrox...)
Affinity DataIC50:  437nMAssay Description:Binding affinity to Leptinotarsa decemlineata EcRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor/Ultraspiracle(Nezara viridula)
Csiro Materials Science And Engineering And Csiro Food And Nutritional Sciences

Curated by ChEMBL
LigandPNGBDBM50226672(CHEMBL255034 | makisterone A)
Affinity DataIC50:  1.38E+3nMAssay Description:Binding affinity to Nezara viridula EcRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEcdysone receptor/Ultraspiracle isoform-A(Aedes aegypti)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50488466(CHEMBL2286418)
Affinity DataEC50:  646nMAssay Description:Agonist activity at Aedes aegypti ecdysone receptor expressed in mammalian cells by reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed