Compile Data Set for Download or QSAR
Report error Found 46 Enz. Inhib. hit(s) with Target = 'Isoform Alpha-1 of Mitogen-activated protein kinase 10 (Alpha-1) 9-402]'
LigandChemical structure of BindingDB Monomer ID 32487BDBM32487(aryl piperidine, 9b)
Affinity DataIC50: 60nMAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32488BDBM32488(aryl piperidine, 9d)
Affinity DataIC50: 80nMAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32494BDBM32494(aryl piperidine, 9j)
Affinity DataIC50: 110nMAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32460BDBM32460(piperazine amide, 4g)
Affinity DataIC50: 160nMpH: 7.0 T: 2°CAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandChemical structure of BindingDB Monomer ID 32469BDBM32469(piperazine amide, 4p)
Affinity DataIC50: 200nMpH: 7.0 T: 2°CAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32490BDBM32490(aryl piperidine, 9f)
Affinity DataIC50: 210nMAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32462BDBM32462(piperazine amide, 4i)
Affinity DataIC50: 250nMpH: 7.0 T: 2°CAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32470BDBM32470(piperazine amide, 4q)
Affinity DataIC50: 290nMpH: 7.0 T: 2°CAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32476BDBM32476(piperazine amide, 6b)
Affinity DataIC50: 310nMpH: 7.0 T: 2°CAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32458BDBM32458(piperazine amide, 6a | piperazine amide, 4e)
Affinity DataIC50: 330nMpH: 7.0 T: 2°CAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32492BDBM32492(aryl piperidine, 9h)
Affinity DataIC50: 350nMAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32489BDBM32489(aryl piperidine, 9e)
Affinity DataIC50: 410nMAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32491BDBM32491(aryl piperidine, 9g)
Affinity DataIC50: 530nMAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32459BDBM32459(piperazine amide, 4f)
Affinity DataIC50: 540nMpH: 7.0 T: 2°CAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32496BDBM32496(aryl piperidine, 9l)
Affinity DataIC50: 620nMAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32466BDBM32466(piperazine amide, 4m)
Affinity DataIC50: 810nMpH: 7.0 T: 2°CAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32456BDBM32456(piperazine amide, 4c)
Affinity DataIC50: 900nMpH: 7.0 T: 2°CAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32461BDBM32461(piperazine amide, 4h)
Affinity DataIC50: 960nMpH: 7.0 T: 2°CAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32493BDBM32493(aryl piperidine, 9i)
Affinity DataIC50: 1.00E+3nMAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32465BDBM32465(piperazine amide, 4l)
Affinity DataIC50: 1.00E+3nMpH: 7.0 T: 2°CAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32463BDBM32463(piperazine amide, 4j)
Affinity DataIC50: 1.10E+3nMpH: 7.0 T: 2°CAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32455BDBM32455(cid_979869 | piperazine amide, 1)
Affinity DataIC50: 1.10E+3nMpH: 7.0 T: 2°CAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32454BDBM32454(piperazine amide, 4b)
Affinity DataIC50: 1.20E+3nMpH: 7.0 T: 2°CAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32458BDBM32458(piperazine amide, 6a | piperazine amide, 4e)
Affinity DataIC50: 1.26E+3nMpH: 7.0 T: 2°CAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32464BDBM32464(piperazine amide, 4k)
Affinity DataIC50: 1.40E+3nMpH: 7.0 T: 2°CAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32477BDBM32477(piperazine amide, 6c)
Affinity DataIC50: 1.80E+3nMpH: 7.0 T: 2°CAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32482BDBM32482(piperazine amide, 6i)
Affinity DataIC50: 2.00E+3nMpH: 7.0 T: 2°CAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32483BDBM32483(piperazine amide, 6j)
Affinity DataIC50: 2.00E+3nMAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32457BDBM32457(piperazine amide, 4d)
Affinity DataIC50: 2.20E+3nMpH: 7.0 T: 2°CAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32478BDBM32478(piperazine amide, 6d)
Affinity DataIC50: 2.30E+3nMpH: 7.0 T: 2°CAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32495BDBM32495(aryl piperidine, 9k)
Affinity DataIC50: 4.80E+3nMAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32479BDBM32479(piperazine amide, 6f)
Affinity DataIC50: 5.00E+3nMpH: 7.0 T: 2°CAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32481BDBM32481(piperazine amide, 6h)
Affinity DataIC50: 5.80E+3nMpH: 7.0 T: 2°CAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32484BDBM32484(piperazine amide, 6k)
Affinity DataIC50: 6.40E+3nMAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32480BDBM32480(piperazine amide, 6g)
Affinity DataIC50: 8.90E+3nMpH: 7.0 T: 2°CAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32453BDBM32453(piperazine amide, 4a)
Affinity DataIC50: 9.90E+3nMpH: 7.0 T: 2°CAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32497BDBM32497(aryl piperidine, 9m)
Affinity DataIC50: 1.10E+4nMAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32472BDBM32472(piperazine amide, 4s)
Affinity DataIC50: 2.00E+4nMpH: 7.0 T: 2°CAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32473BDBM32473(piperazine amide, 4t)
Affinity DataIC50: 2.00E+4nMpH: 7.0 T: 2°CAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32474BDBM32474(piperazine amide, 4u)
Affinity DataIC50: 2.00E+4nMpH: 7.0 T: 2°CAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32498BDBM32498(aryl piperidine, 9n)
Affinity DataIC50: 2.00E+4nMAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32467BDBM32467(piperazine amide, 4n)
Affinity DataIC50: 2.00E+4nMpH: 7.0 T: 2°CAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32468BDBM32468(piperazine amide, 4o)
Affinity DataIC50: 2.00E+4nMpH: 7.0 T: 2°CAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32485BDBM32485(piperazine amide, 6l)
Affinity DataIC50: 2.00E+4nMAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32486BDBM32486(piperazine amide, 6m)
Affinity DataIC50: 2.00E+4nMAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 32471BDBM32471(piperazine amide, 4r)
Affinity DataIC50: 2.00E+4nMpH: 7.0 T: 2°CAssay Description:Biochemical IC50s for JNK were determined using HTRF. In each assay the phosphor-Thr71-ATF-2 product was detected using a Europium-cryptate labeled a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2009
Entry Details Article
PubMed