Report error Found 156 Enz. Inhib. hit(s) with Target = 'Pancreatic alpha-amylase'
Displayed 1 to 50 (of 156 total ) | Next | Last >>
Affinity DataEC50: 0.0500nMAssay Description:Tested in vitro for amylase release from rat pancreatic aciniMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Tested in vitro for inhibition of amylase release from rat pancreatic aciniMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Tested in vitro for inhibition of amylase release from rat pancreatic aciniMore data for this Ligand-Target Pair
Affinity DataKi: 1nMpH: 7.0Assay Description:The release of 2-chloro-4-nitrophenol resulting from the HPA-catalyzed hydrolysis of 2-chloro-4-nitrophenyl a-maltotrioside (CNPG3) was monitored at ...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Tested in vitro for inhibition of amylase release from rat pancreatic aciniMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMpH: 7.0Assay Description:The release of 2-chloro-4-nitrophenol resulting from the HPA-catalyzed hydrolysis of 2-chloro-4-nitrophenyl a-maltotrioside (CNPG3) was monitored at ...More data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Tested in vitro for amylase release from rat pancreatic acini (percent of secretion)More data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Tested in vitro for amylase release from rat pancreatic acini (percent of secretion)More data for this Ligand-Target Pair
Affinity DataEC50: 6nMAssay Description:Tested in vitro for amylase release from rat pancreatic acini (percent of secretion)More data for this Ligand-Target Pair
Affinity DataKi: 7nMpH: 7.0Assay Description:The release of 2-chloro-4-nitrophenol resulting from the HPA-catalyzed hydrolysis of 2-chloro-4-nitrophenyl a-maltotrioside (CNPG3) was monitored at ...More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Tested in vitro for inhibition of amylase release from rat pancreatic aciniMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Competitive inhibition of human pancreatic alpha-amylase by double reciprocal plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 8.10nM ΔG°: -47.0kJ/moleT: 2°CAssay Description:Inhibitor concentrations varied from 0.25 to 5 times the Ki value in 50 mM sodium phosphate, 100 mM sodium chloride buffer, pH 7.0, at 30 °C. 2-Chlor...More data for this Ligand-Target Pair
Affinity DataIC50: 8.5nMpH: 7.0Assay Description:After kinetic analysis with HPA, piHA-Dm was tested as an inhibitor of ten additional enzymes. The conditions are listed as follows: Agrobacterium fa...More data for this Ligand-Target Pair
Affinity DataKi: 9.10nM ΔG°: -46.7kJ/moleT: 2°CAssay Description:Inhibitor concentrations varied from 0.25 to 5 times the Ki value in 50 mM sodium phosphate, 100 mM sodium chloride buffer, pH 7.0, at 30 °C. 2-Chlor...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of the release of Alpha-amylase from rat pancreatic acinar cells.More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Inhibition of human pancreatic alpha-amylaseMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Inhibition of human pancreatic alpha-amylaseMore data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataKi: 14nMAssay Description:Inhibition of human pancreatic alpha-amylase expressed in Pichia pastoris using amylase as substrate preincubated with substrate for 10 mins followed...More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Inhibition of human pancreatic alpha-amylase expressed in Pichia pastoris using amylase as substrate preincubated with substrate for 10 mins followed...More data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Tested in vitro for amylase release from rat pancreatic acini (percent of secretion)More data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Tested in vitro for amylase release from rat pancreatic acini (percent of secretion)More data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibition of the release of Alpha-amylase from rat pancreatic acinar cells.More data for this Ligand-Target Pair
Affinity DataKi: 21.3nM ΔG°: -44.5kJ/moleT: 2°CAssay Description:Inhibitor concentrations varied from 0.25 to 5 times the Ki value in 50 mM sodium phosphate, 100 mM sodium chloride buffer, pH 7.0, at 30 °C. 2-Chlor...More data for this Ligand-Target Pair
Affinity DataEC50: 22nMAssay Description:Tested in vitro for amylase release from rat pancreatic acini (% of amylase secretion at 1 mM)More data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Inhibition of human pancreatic alpha-amylase expressed in Pichia pastoris using amylase as substrate preincubated with substrate for 10 mins followed...More data for this Ligand-Target Pair
Affinity DataKi: 42.4nM ΔG°: -42.8kJ/moleT: 2°CAssay Description:Inhibitor concentrations varied from 0.25 to 5 times the Ki value in 50 mM sodium phosphate, 100 mM sodium chloride buffer, pH 7.0, at 30 °C. 2-Chlor...More data for this Ligand-Target Pair
Affinity DataIC50: 46nMAssay Description:Inhibition of the release of Alpha-amylase from rat pancreatic acinar cells.More data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Tested in vitro for amylase release from rat pancreatic acini (percent of secretion)More data for this Ligand-Target Pair
Affinity DataIC50: 52nMAssay Description:Inhibition of the release of Alpha-amylase from rat pancreatic acinar cells.More data for this Ligand-Target Pair
Affinity DataKi: 75nMAssay Description:Inhibition of human pancreatic alpha-amylaseMore data for this Ligand-Target Pair
Affinity DataKi: 79.3nM ΔG°: -41.2kJ/moleT: 2°CAssay Description:Inhibitor concentrations varied from 0.25 to 5 times the Ki value in 50 mM sodium phosphate, 100 mM sodium chloride buffer, pH 7.0, at 30 °C. 2-Chlor...More data for this Ligand-Target Pair
Affinity DataKi: 93.3nM ΔG°: -40.8kJ/moleT: 2°CAssay Description:Inhibitor concentrations varied from 0.25 to 5 times the Ki value in 50 mM sodium phosphate, 100 mM sodium chloride buffer, pH 7.0, at 30 °C. 2-Chlor...More data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Inhibition of the release of Alpha-amylase from rat pancreatic acinar cells.More data for this Ligand-Target Pair
Affinity DataIC50: 380nMAssay Description:Inhibition of porcine pancreatic alpha-amylase using 1% starch as substrate preincubated for 10 mins followed by substrate addition and measured afte...More data for this Ligand-Target Pair
Affinity DataIC50: 380nMAssay Description:Inhibition of the release of Alpha-amylase from rat pancreatic acinar cells.More data for this Ligand-Target Pair
Affinity DataIC50: 590nMAssay Description:Inhibition of porcine pancreatic alpha-amylase using starch as substrate incubated for 10 mins by absorbance based assayMore data for this Ligand-Target Pair
Affinity DataKi: 730nM ΔG°: -35.6kJ/moleT: 2°CAssay Description:Inhibitor concentrations varied from 0.25 to 5 times the Ki value in 50 mM sodium phosphate, 100 mM sodium chloride buffer, pH 7.0, at 30 °C. 2-Chlor...More data for this Ligand-Target Pair
Affinity DataKi: 1.25E+3nMAssay Description:Inhibition of human pancreatic alpha-amylase expressed in Pichia pastoris using amylase as substrate preincubated with substrate for 10 mins followed...More data for this Ligand-Target Pair
Affinity DataIC50: 1.35E+3nMAssay Description:Inhibition of porcine pancreatic alpha-amylase using starch as substrate preincubated for 10 mins followed by substrate addition measured after 10 mi...More data for this Ligand-Target Pair
Affinity DataIC50: 1.57E+3nMAssay Description:Inhibition of porcine pancreatic alpha-amylase using starch as substrate preincubated for 10 mins followed by substrate addition measured after 10 mi...More data for this Ligand-Target Pair
Affinity DataIC50: 1.66E+3nMAssay Description:Inhibition of porcine pancreatic alpha-amylase using 1% starch as substrate preincubated for 10 mins followed by substrate addition and measured afte...More data for this Ligand-Target Pair
Affinity DataIC50: 1.66E+3nMAssay Description:Inhibition of porcine pancreatic alpha-amylase using 1% starch as substrate preincubated for 10 mins followed by substrate addition and measured afte...More data for this Ligand-Target Pair
Affinity DataIC50: 2.06E+3nMAssay Description:Inhibition of porcine pancreatic alpha-amylase using starch as substrate preincubated for 10 mins followed by substrate addition measured after 10 mi...More data for this Ligand-Target Pair
Affinity DataIC50: 2.12E+3nMAssay Description:Inhibition of porcine pancreatic alpha-amylase using starch as substrate preincubated for 10 mins followed by substrate addition measured after 10 mi...More data for this Ligand-Target Pair
Affinity DataKi: 2.24E+3nM ΔG°: -32.8kJ/moleT: 2°CAssay Description:Inhibitor concentrations varied from 0.25 to 5 times the Ki value in 50 mM sodium phosphate, 100 mM sodium chloride buffer, pH 7.0, at 30 °C. 2-Chlor...More data for this Ligand-Target Pair
Affinity DataIC50: 2.35E+3nMAssay Description:Inhibition of porcine pancreatic alpha-amylase using starch as substrate preincubated for 10 mins followed by substrate addition measured after 10 mi...More data for this Ligand-Target Pair
Affinity DataIC50: 2.59E+3nMAssay Description:Inhibition of human pancreatic alpha-amylase expressed in Pichia pastoris using amylase as substrate preincubated with substrate for 10 mins followed...More data for this Ligand-Target Pair
Affinity DataIC50: 2.67E+3nMAssay Description:Inhibition of porcine pancreatic alpha-amylase using starch as substrate preincubated for 10 mins followed by substrate addition measured after 10 mi...More data for this Ligand-Target Pair
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of the release of Alpha-amylase from rat pancreatic acinar cells.More data for this Ligand-Target Pair