Compile Data Set for Download or QSAR
Report error Found 218 Enz. Inhib. hit(s) with Target = 'Solute carrier family 22 member 6'
TargetSolute carrier family 22 member 6(Human)
Kyorin University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350468BDBM50350468(CEFAMANDOLE)
Affinity DataKi:  30nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in OAT1-expressing S2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSolute carrier family 22 member 6(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206441BDBM50206441(2-(2,4,5,7-tetrabromo-3-hydroxy-6-oxo-6H-xanthen-9...)
Affinity DataKi:  89nMAssay Description:Inhibition of mouse Oat1-mediated [3H]PAH uptake in Xenopus oocytes after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetSolute carrier family 22 member 6(Human)
Kyorin University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370587BDBM50370587(CEFAZOLIN)
Affinity DataKi:  180nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in OAT1-expressing S2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSolute carrier family 22 member 6(Human)
Kyorin University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50390999BDBM50390999(CEFOPERAZONE)
Affinity DataKi:  210nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in OAT1-expressing S2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSolute carrier family 22 member 6(Human)
Kyorin University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 82898BDBM82898(SMR000386987 | MLS001048966 | (6R,7R)-3-(acetyloxy...)
Affinity DataKi:  220nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in OAT1-expressing S2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSolute carrier family 22 member 6(Human)
Kyorin University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50049707BDBM50049707((6R,7R)-7-{2-(2-Amino-thiazol-4-yl)-2-[(Z)-methoxy...)
Affinity DataKi:  230nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in OAT1-expressing S2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSolute carrier family 22 member 6(Human)
Kyorin University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 4078BDBM4078(Elagic Acid | CHEMBL6246 | 6,7,13,14-tetrahydroxy-...)
Affinity DataIC50: 270nMAssay Description:TP_TRANSPORTER: inhibition of ochratoxin A uptake (ochratoxin A / 1uM) in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSolute carrier family 22 member 6(Rat)
University of Rochester School of Medicine and Dentistry

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50485601BDBM50485601(CHEMBL2075007)
Affinity DataKi:  400nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMed
TargetSolute carrier family 22 member 6(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50270022BDBM50270022(hexanedioic acid, ion(2-) | hexanedioate | adipate...)
Affinity DataKi:  410nMAssay Description:Inhibition of mouse Oat1-mediated [3H]PAH uptake in Xenopus oocytes after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetSolute carrier family 22 member 6(Rat)
University of Rochester School of Medicine and Dentistry

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50022271BDBM50022271(2-(3-benzoylphenyl)propanoic acid | 2-(3-Benzoylph...)
Affinity DataIC50: 500nMAssay Description:TP_TRANSPORTER: inhibition of MTX uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSolute carrier family 22 member 6(Human)
Kyorin University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350473BDBM50350473(Aliporina | CEFALORIDINE)
Affinity DataKi:  740nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in OAT1-expressing S2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSolute carrier family 22 member 6(Human)
Kyorin University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50240510BDBM50240510(CHEMBL898 | DIFLUNISAL)
Affinity DataIC50: 850nMAssay Description:TP_TRANSPORTER: inhibition of Adefovir uptake in OAT1-expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details
PubMed
TargetSolute carrier family 22 member 6(Rat)
University of Rochester School of Medicine and Dentistry

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50485602BDBM50485602(CHEMBL2075010)
Affinity DataKi:  1.10E+3nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMed
TargetSolute carrier family 22 member 6(Human)
Kyorin University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50022271BDBM50022271(2-(3-benzoylphenyl)propanoic acid | 2-(3-Benzoylph...)
Affinity DataIC50: 1.30E+3nMAssay Description:TP_TRANSPORTER: inhibition of Adefovir uptake in OAT1-expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details
PubMed
TargetSolute carrier family 22 member 6(Human)
Kyorin University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50022271BDBM50022271(2-(3-benzoylphenyl)propanoic acid | 2-(3-Benzoylph...)
Affinity DataIC50: 1.40E+3nMAssay Description:TP_TRANSPORTER: inhibition of 6-Carboxyfluorescein uptake in OAT1-expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetSolute carrier family 22 member 6(Human)
Kyorin University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50074922BDBM50074922(2-(2-fluoro-[1,1'-biphenyl-4-yl])propanoic acid | ...)
Affinity DataIC50: 1.50E+3nMAssay Description:TP_TRANSPORTER: inhibition of Adefovir uptake in OAT1-expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details
PubMed
TargetSolute carrier family 22 member 6(Rat)
University of Rochester School of Medicine and Dentistry

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50012957BDBM50012957(1-((p-(2-(5-chloro-o-anisamido)ethyl)phenyl)sulfon...)
Affinity DataKi:  1.60E+3nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSolute carrier family 22 member 6(Rat)
University of Rochester School of Medicine and Dentistry

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50485603BDBM50485603(CHEBI:7426 | CHEMBL2074738)
Affinity DataKi:  1.90E+3nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMed
TargetSolute carrier family 22 member 6(Rat)
University of Rochester School of Medicine and Dentistry

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339185BDBM50339185((2S)-2-(6-methoxynaphthalen-2-yl)propanoic acid | ...)
Affinity DataKi:  2.00E+3nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details
PubMed
TargetSolute carrier family 22 member 6(Human)
Kyorin University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50158460BDBM50158460(cid_2333 | Benzbromarone | 3,5-dibromo-4-hydroxyph...)
Affinity DataIC50: 2.12E+3nMAssay Description:Inhibition of OAT1 (unknown origin) transfected in HEK293 cells assessed as inhibition of 6-CFL uptake preincubated for 30 mins followed by 6-CFL add...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetSolute carrier family 22 member 6(Rat)
University of Rochester School of Medicine and Dentistry

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50420231BDBM50420231(CHEMBL2074600)
Affinity DataKi:  2.74E+3nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in Oat1-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSolute carrier family 22 member 6(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50143424BDBM50143424(2-(3-hydroxy-6-oxo-6H-xanthen-9-yl)benzoic acid | ...)
Affinity DataKi:  2.95E+3nMAssay Description:Inhibition of mouse Oat1-mediated [3H]PAH uptake in Xenopus oocytes after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetSolute carrier family 22 member 6(Human)
Kyorin University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50133599BDBM50133599(CHEMBL119625 | YM-872 | (7-Imidazol-1-yl-6-nitro-2...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human OAT1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSolute carrier family 22 member 6(Human)
Kyorin University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 17638BDBM17638(indometacin | Indocin | 2-{1-[(4-chlorophenyl)carb...)
Affinity DataIC50: 3.00E+3nMAssay Description:TP_TRANSPORTER: inhibition of Adefovir uptake in OAT1-expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details
PubMed
TargetSolute carrier family 22 member 6(Human)
Kyorin University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50335523BDBM50335523(Claforan | Kefotex | cefotaxim | cefotaxime | (6R,...)
Affinity DataKi:  3.13E+3nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in OAT1-expressing S2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSolute carrier family 22 member 6(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 35847BDBM35847(DINOPROSTONE | [3H]Prostaglandin E2 | prostaglandi...)
Affinity DataKi:  3.40E+3nMAssay Description:Inhibition of mouse Oat1-mediated [3H]PAH uptake in Xenopus oocytes after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetSolute carrier family 22 member 6(Rat)
University of Rochester School of Medicine and Dentistry

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50009859BDBM50009859((RS)-ibuprofen | CHEMBL521 | 2-(4-isobutylphenyl)p...)
Affinity DataKi:  3.50E+3nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details
PubMed
TargetSolute carrier family 22 member 6(Human)
Kyorin University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50537496BDBM50537496(CHEMBL4527448)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of OAT1 (unknown origin) expressed in HEK293 cells assessed as reduction in 6-CF uptake measured after 5 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSolute carrier family 22 member 6(Human)
Kyorin University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13066BDBM13066({2-[(2,6-dichlorophenyl)amino]phenyl}acetic acid |...)
Affinity DataIC50: 4.00E+3nMAssay Description:TP_TRANSPORTER: inhibition of Adefovir uptake in OAT1-expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details
PubMed
TargetSolute carrier family 22 member 6(Rat)
University of Rochester School of Medicine and Dentistry

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 17638BDBM17638(indometacin | Indocin | 2-{1-[(4-chlorophenyl)carb...)
Affinity DataKi:  4.20E+3nMAssay Description:TP_TRANSPORTER: inhibition of MTX uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSolute carrier family 22 member 6(Human)
Kyorin University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206509BDBM50206509(CHEMBL897 | 4-Dipropylsulfamoyl-benzoic acid(probe...)
Affinity DataKi:  4.30E+3nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in OAT1-expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSolute carrier family 22 member 6(Human)
Kyorin University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50537500BDBM50537500(CHEMBL4562825)
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of OAT1 (unknown origin) expressed in HEK293 cells assessed as reduction in 6-CF uptake measured after 5 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSolute carrier family 22 member 6(Human)
Kyorin University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206509BDBM50206509(CHEMBL897 | 4-Dipropylsulfamoyl-benzoic acid(probe...)
Affinity DataKi:  4.41E+3nMAssay Description:TP_TRANSPORTER: inhibition of Ochratoxin A uptake in OAT1-expressing S2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSolute carrier family 22 member 6(Human)
Kyorin University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50158460BDBM50158460(cid_2333 | Benzbromarone | 3,5-dibromo-4-hydroxyph...)
Affinity DataIC50: 4.60E+3nMAssay Description:TP_TRANSPORTER: inhibition of Urate uptake (Urate: 300 uM) in OAT1-expressing S2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMed
TargetSolute carrier family 22 member 6(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50009859BDBM50009859((RS)-ibuprofen | CHEMBL521 | 2-(4-isobutylphenyl)p...)
Affinity DataKi:  4.70E+3nMAssay Description:Inhibition of mouse Oat1-mediated [3H]PAH uptake in Xenopus oocytes after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetSolute carrier family 22 member 6(Human)
Kyorin University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50485550BDBM50485550(CHEBI:17859 | Glutarate)
Affinity DataIC50: 4.90E+3nMAssay Description:TP_TRANSPORTER: inhibition of 6-Carboxyfluorescein uptake in OAT1-expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetSolute carrier family 22 member 6(Human)
Kyorin University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50485608BDBM50485608(CHEBI:28837 | Caprylic acid | EDENOR C 8-98-100 | ...)
Affinity DataKi:  5.41E+3nMAssay Description:TP_TRANSPORTER: inhibition of Ochratoxin A uptake in OAT1-expressing S2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMed
TargetSolute carrier family 22 member 6(Rat)
University of Rochester School of Medicine and Dentistry

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 25903BDBM25903(Fordiuran | Burinex | cid_2471 | 3-(butylamino)-4-...)
Affinity DataKi:  5.50E+3nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details
PubMed
TargetSolute carrier family 22 member 6(Human)
Kyorin University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339185BDBM50339185((2S)-2-(6-methoxynaphthalen-2-yl)propanoic acid | ...)
Affinity DataIC50: 5.80E+3nMAssay Description:TP_TRANSPORTER: inhibition of Adefovir uptake in OAT1-expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details
PubMed
TargetSolute carrier family 22 member 6(Human)
Kyorin University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50344964BDBM50344964(Betamipron | N-(phenylcarbonyl)-beta-alanine | CHE...)
Affinity DataIC50: 6.00E+3nMAssay Description:TP_TRANSPORTER: inhibition of Adefovir uptake in OAT1-expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details
PubMed
TargetSolute carrier family 22 member 6(Human)
Kyorin University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50270006BDBM50270006(2-(4-aminobenzamido)acetate | AMINOHIPPURATE)
Affinity DataKi:  6.02E+3nMAssay Description:Inhibition of human Oat1 expressed in Drosophila S2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2013
Entry Details Article
PubMed
TargetSolute carrier family 22 member 6(Human)
Kyorin University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50240008BDBM50240008(CHEBI:104011 | Aminohippuric Acid | PAHA | Para-Am...)
Affinity DataKi:  6.02E+3nMAssay Description:TP_TRANSPORTER: inhibition of Ochratoxin A uptake in OAT1-expressing S2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSolute carrier family 22 member 6(Human)
Kyorin University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350467BDBM50350467(BL-S578 | Cefadrops | CEFADROXIL)
Affinity DataKi:  6.14E+3nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in OAT1-expressing S2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSolute carrier family 22 member 6(Human)
Kyorin University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50637872BDBM50637872(CHEMBL5542977)
Affinity DataIC50: 6.19E+3nMAssay Description:Inhibition of human OAT1 expressed in MDCK-II cells using 6-carboxyfluorescein as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSolute carrier family 22 member 6(Human)
Kyorin University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206509BDBM50206509(CHEMBL897 | 4-Dipropylsulfamoyl-benzoic acid(probe...)
Affinity DataIC50: 6.30E+3nMAssay Description:TP_TRANSPORTER: inhibition of 6-Carboxyfluorescein uptake in OAT1-expressing CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSolute carrier family 22 member 6(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50269998BDBM50269998((S)-2-((R)-5-chloro-8-hydroxy-3-methyl-1-oxoisochr...)
Affinity DataKi:  6.31E+3nMAssay Description:Inhibition of mouse Oat1-mediated [3H]PAH uptake in Xenopus oocytes after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetSolute carrier family 22 member 6(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206509BDBM50206509(CHEMBL897 | 4-Dipropylsulfamoyl-benzoic acid(probe...)
Affinity DataKi:  6.31E+3nMAssay Description:Inhibition of mouse Oat1-mediated [3H]PAH uptake in Xenopus oocytes after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSolute carrier family 22 member 6(Human)
Kyorin University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50206509BDBM50206509(CHEMBL897 | 4-Dipropylsulfamoyl-benzoic acid(probe...)
Affinity DataIC50: 6.51E+3nMAssay Description:Experimental results: The compounds had no obvious inhibitory effect on the drug transporter OAT3, and when the compounds were used clinically in com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2024
Entry Details
US Patent
PDB3D3D Structure (crystal)
TargetSolute carrier family 22 member 6(Mouse)
University of California

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50270021BDBM50270021(glutarate(2-) | pentanedioate | glutarate)
Affinity DataKi:  6.70E+3nMAssay Description:Inhibition of mouse Oat1-mediated [3H]PAH uptake in Xenopus oocytes after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetSolute carrier family 22 member 6(Human)
Kyorin University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50538736BDBM50538736(CHEMBL4640580)
Affinity DataKi:  7.20E+3nMAssay Description:Inhibition of human OAT1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
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