Compile Data Set for Download or QSAR
Report error Found 75 Enz. Inhib. hit(s) with Target = 'Stromelysin-3'
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50480363BDBM50480363(CHEMBL449897)
Affinity DataIC50: 0.0250nMAssay Description:Cytotoxicity against human NB-1 cells by MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50480365BDBM50480365(CHEMBL466909)
Affinity DataIC50: 0.0280nMAssay Description:Cytotoxicity against human NB-1 cells by MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50404889BDBM50404889(CHEMBL303714)
Affinity DataIC50: 0.0280nMAssay Description:Cytotoxicity against human NB-1 cells by MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50480366BDBM50480366(CHEMBL513819)
Affinity DataIC50: 0.0290nMAssay Description:Cytotoxicity against human NB-1 cells by MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50480364BDBM50480364(CHEMBL468539)
Affinity DataIC50: 0.0320nMAssay Description:Cytotoxicity against human NB-1 cells by MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50480360BDBM50480360(CHEMBL466908)
Affinity DataIC50: 0.0320nMAssay Description:Cytotoxicity against human NB-1 cells by MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50480362BDBM50480362(CHEMBL466114)
Affinity DataIC50: 0.0330nMAssay Description:Cytotoxicity against human NB-1 cells by MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50480367BDBM50480367(CHEMBL468747)
Affinity DataIC50: 0.0330nMAssay Description:Cytotoxicity against human NB-1 cells by MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50480359BDBM50480359(CHEMBL466907)
Affinity DataIC50: 0.0400nMAssay Description:Cytotoxicity against human NB-1 cells by MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50480361BDBM50480361(CHEMBL511905)
Affinity DataIC50: 0.0430nMAssay Description:Cytotoxicity against human NB-1 cells by MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetStromelysin-3(Human)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50265077BDBM50265077((S)-3-((S)-1-amino-3-(1H-indol-3-yl)-1-oxopropan-2...)
Affinity DataKi:  0.230nMAssay Description:Inhibition of MMP11More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078935BDBM50078935((2-{N-[1-Carbamoyl-2-(1H-indol-3-yl)-ethyl]-hydraz...)
Affinity DataKi:  0.900nMAssay Description:Binding affinity against matrix metalloprotease-11.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078950BDBM50078950((2-{N-[1-Carbamoyl-2-(1H-indol-3-yl)-ethyl]-hydraz...)
Affinity DataKi:  1.5nMAssay Description:Binding affinity against matrix metalloprotease-11.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078947BDBM50078947((1-Benzyloxycarbonylamino-2-phenyl-ethyl)-[2-[1-ca...)
Affinity DataKi:  2nMAssay Description:Binding affinity against matrix metalloprotease-11.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078945BDBM50078945((2-{N-[1-Carbamoyl-2-(1H-indol-3-yl)-ethyl]-hydraz...)
Affinity DataKi:  3.80nMAssay Description:Binding affinity against matrix metalloprotease-11.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078932BDBM50078932((2-{N-[1-Carbamoyl-2-(1H-indol-3-yl)-ethyl]-hydraz...)
Affinity DataKi:  4.20nMAssay Description:Binding affinity against matrix metalloprotease-11.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50362781BDBM50362781(CHEMBL1738797 | US9126931, 366 | Alectinib | 12565...)
Affinity DataIC50: 4.5nMAssay Description:Antiproliferative activity against human NB1 cells harbouring ALK by CellTiter-Glo luminescent cell viability assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50138684BDBM50138684((1-Benzyloxycarbonylamino-2-phenyl-ethyl)-{2-[1-ca...)
Affinity DataKi:  5nMAssay Description:Inhibition of Matrix metalloprotease-11More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078938BDBM50078938((2-{N-[1-Carbamoyl-2-(1H-indol-3-yl)-ethyl]-hydraz...)
Affinity DataKi:  5nMAssay Description:Binding affinity against matrix metalloprotease-11.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078930BDBM50078930((1-Benzyloxycarbonylamino-2-phenyl-ethyl)-{2-[(R)-...)
Affinity DataKi:  5nMAssay Description:Binding affinity against matrix metalloprotease-11.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-3(Human)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393211BDBM50393211(CHEMBL2153737)
Affinity DataKi:  5nMAssay Description:Inhibition of MMP-11More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078951BDBM50078951([1-(2-Benzyloxy-acetylamino)-2-phenyl-ethyl]-{2-[1...)
Affinity DataKi:  5nMAssay Description:Binding affinity against matrix metalloprotease-11.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-3(Human)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50138684BDBM50138684((1-Benzyloxycarbonylamino-2-phenyl-ethyl)-{2-[1-ca...)
Affinity DataKi:  5nMAssay Description:Binding affinity to MMP11More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 22984BDBM22984(Adriamycin | (8S,10S)-10-{[(2R,4S,5S,6S)-4-amino-5...)
Affinity DataIC50: 5.15nMAssay Description:Cytotoxicity against human NB-1 cells by MTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078941BDBM50078941([1-(2-Benzyloxycarbonylamino-4-methyl-pentanoylami...)
Affinity DataKi:  6nMAssay Description:Binding affinity against matrix metalloprotease-11.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078946BDBM50078946([1-(2-Benzyloxycarbonylamino-propionylamino)-2-phe...)
Affinity DataKi:  8nMAssay Description:Binding affinity against matrix metalloprotease-11.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078933BDBM50078933((1-Benzyloxycarbonylamino-2-phenyl-ethyl)-{2-[1-ca...)
Affinity DataKi:  8.80nMAssay Description:Binding affinity against matrix metalloprotease-11.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078929BDBM50078929((2-{N-[1-Carbamoyl-2-(1H-indol-3-yl)-ethyl]-hydraz...)
Affinity DataKi:  10nMAssay Description:Binding affinity against matrix metalloprotease-11.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078948BDBM50078948((1-Benzyloxycarbonylamino-2-phenyl-ethyl)-{2-[1-ca...)
Affinity DataKi:  12nMAssay Description:Binding affinity against matrix metalloprotease-11.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078928BDBM50078928((2-{N-[1-Carbamoyl-2-(1H-indol-3-yl)-ethyl]-hydraz...)
Affinity DataKi:  15nMAssay Description:Binding affinity against matrix metalloprotease-11.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078942BDBM50078942({3-Benzyloxy-2-[1-carbamoyl-2-(1H-indol-3-yl)-ethy...)
Affinity DataKi:  16nMAssay Description:Binding affinity against matrix metalloprotease-11.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078943BDBM50078943((1-Acetylamino-2-phenyl-ethyl)-{2-[1-carbamoyl-2-(...)
Affinity DataKi:  20nMAssay Description:Binding affinity against matrix metalloprotease-11.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078949BDBM50078949((1-Benzyloxycarbonylamino-2-phenyl-ethyl)-{2-[1-ca...)
Affinity DataKi:  22nMAssay Description:Binding affinity against matrix metalloprotease-11.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078936BDBM50078936({2-[(2-Amino-1-carbamoyl-ethyl)-(2,4-dinitro-pheny...)
Affinity DataKi:  27nMAssay Description:Binding affinity against matrix metalloprotease-11.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078953BDBM50078953((1-Benzyloxycarbonylamino-2-phenyl-ethyl)-{2-[1-ca...)
Affinity DataKi:  33nMAssay Description:Binding affinity against matrix metalloprotease-11.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078939BDBM50078939((1-Benzyloxycarbonylamino-2-phenyl-ethyl)-{2-[1-ca...)
Affinity DataKi:  34nMAssay Description:Binding affinity against matrix metalloprotease-11.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078937BDBM50078937((1-Benzyloxycarbonylamino-ethyl)-{3-benzylsulfanyl...)
Affinity DataKi:  36nMAssay Description:Binding affinity against matrix metalloprotease-11.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078931BDBM50078931((1-Benzyloxycarbonylamino-ethyl)-{2-[1-carbamoyl-2...)
Affinity DataKi:  51nMAssay Description:Binding affinity against matrix metalloprotease-11.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078940BDBM50078940((1-Benzyloxycarbonylamino-2-phenyl-ethyl)-{2-[1-ca...)
Affinity DataKi:  74nMAssay Description:Binding affinity against matrix metalloprotease-11.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078954BDBM50078954((1-Benzyloxycarbonylamino-ethyl)-{2-[1-carbamoyl-2...)
Affinity DataKi:  100nMAssay Description:Binding affinity against matrix metalloprotease-11.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50138683BDBM50138683((1-Benzyloxycarbonylamino-2-phenyl-ethyl)-{3-(2-br...)
Affinity DataKi:  110nMAssay Description:Inhibition of Matrix metalloprotease-11More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078952BDBM50078952({3-Benzyloxy-2-[1-carbamoyl-2-(1H-indol-3-yl)-ethy...)
Affinity DataKi:  175nMAssay Description:Binding affinity against matrix metalloprotease-11.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50138685BDBM50138685((1-Benzyloxycarbonylamino-2-phenyl-ethyl)-[2-[1-ca...)
Affinity DataKi:  230nMAssay Description:Inhibition of Matrix metalloprotease-11More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078944BDBM50078944((1-Benzyloxycarbonylamino-ethyl)-{2-[1-carbamoyl-2...)
Affinity DataKi:  350nMAssay Description:Binding affinity against matrix metalloprotease-11.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50138686BDBM50138686((1-Benzyloxycarbonylamino-2-phenyl-ethyl)-[2-[1-ca...)
Affinity DataKi:  410nMAssay Description:Inhibition of Matrix metalloprotease-11More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-3(Human)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393207BDBM50393207(CHEMBL2153738)
Affinity DataKi:  410nMAssay Description:Inhibition of MMP-11More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078955BDBM50078955((1-Benzyloxycarbonylamino-2-phenyl-ethyl)-{2-[1-ca...)
Affinity DataKi:  2.67E+3nMAssay Description:Binding affinity against matrix metalloprotease-11.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-3(Human)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50302107BDBM50302107(Grassystatin A | CHEMBL567893)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of MMP11 catalytic domain after 10 to 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetStromelysin-3(Mouse)
National Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50615275BDBM50615275(CHEMBL5282240)
Affinity DataIC50: 1.02E+4nMAssay Description:Cytotoxicity against human NB1 cells measured after 8 daysMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetStromelysin-3(Human)
University of Athens

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50265078BDBM50265078((4S)-5-amino-4-((2S)-2-((2S)-3-((4-bromophenyl)(hy...)
Affinity DataKi:  1.84E+4nMAssay Description:Inhibition of MMP11More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
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