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Found 100 with Last Name = 'allaoa' and Initial = 'a'
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Memorial Sloan Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50531606(CHEMBL4514672)
Affinity DataKi:  8.60nMAssay Description:Displacement of [3H]Pentazocine from guinea pig sigma-1 receptor by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)TBA
LigandPNGBDBM50609010(CHEMBL5276728)
Affinity DataKi:  34nMAssay Description:Displacement of [125]IBNtxA from mouse MOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50609010(CHEMBL5276728)
Affinity DataKi:  49nMAssay Description:Displacement of [125]IBNtxA from mouse DOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Memorial Sloan Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50531605(CHEMBL4552298)
Affinity DataKi:  58nMAssay Description:Displacement of [3H]Pentazocine from guinea pig sigma-1 receptor by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)TBA
LigandPNGBDBM50519927(CHEMBL4546925)
Affinity DataKi:  79nMAssay Description:Displacement of [125]IBNtxA from mouse MOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetKappa-type opioid receptor(Mus musculus (Mouse))TBA
LigandPNGBDBM50609010(CHEMBL5276728)
Affinity DataKi:  125nMAssay Description:Displacement of [125]IBNtxA from mouse KOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMu-type opioid receptor(MOUSE)TBA
LigandPNGBDBM50474151(CHEMBL292521)
Affinity DataKi:  216nMAssay Description:Displacement of [125]IBNtxA from mouse MOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Memorial Sloan Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50531606(CHEMBL4514672)
Affinity DataKi:  231nMAssay Description:Displacement of [3H]LSD from human 5-HT2B receptor expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
Memorial Sloan Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50531604(CHEMBL4562437)
Affinity DataKi:  546nMAssay Description:Binding affinity to human histamine 2 receptor expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)TBA
LigandPNGBDBM50566316(CHEMBL4859858)
Affinity DataKi:  578nMAssay Description:Displacement of [125]IBNtxA from mouse MOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKappa-type opioid receptor(Mus musculus (Mouse))TBA
LigandPNGBDBM50519927(CHEMBL4546925)
Affinity DataKi:  649nMAssay Description:Displacement of [125]IBNtxA from mouse KOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(MOUSE)TBA
LigandPNGBDBM50566317(CHEMBL4848517)
Affinity DataKi:  666nMAssay Description:Displacement of [125]IBNtxA from mouse MOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
Memorial Sloan Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50531606(CHEMBL4514672)
Affinity DataKi:  696nMAssay Description:Displacement of [3H]DTG from sigma-2 receptor in rat PC12 cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Memorial Sloan Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50531607(CHEMBL4472251)
Affinity DataKi:  742nMAssay Description:Displacement of [3H]LSD from human 5-HT2B receptor expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
Memorial Sloan Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50531606(CHEMBL4514672)
Affinity DataKi:  823nMAssay Description:Binding affinity to human histamine 2 receptor expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Memorial Sloan Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50531604(CHEMBL4562437)
Affinity DataKi:  840nMAssay Description:Displacement of [3H]LSD from human 5-HT2B receptor expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Mus musculus (Mouse))TBA
LigandPNGBDBM50566317(CHEMBL4848517)
Affinity DataKi:  883nMAssay Description:Displacement of [125]IBNtxA from mouse KOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Memorial Sloan Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50531604(CHEMBL4562437)
Affinity DataKi:  993nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50519927(CHEMBL4546925)
Affinity DataKi:  1.15E+3nMAssay Description:Displacement of [125]IBNtxA from mouse DOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetKappa-type opioid receptor(Mus musculus (Mouse))TBA
LigandPNGBDBM50474151(CHEMBL292521)
Affinity DataKi:  1.18E+3nMAssay Description:Displacement of [125]IBNtxA from mouse KOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetKappa-type opioid receptor(Mus musculus (Mouse))TBA
LigandPNGBDBM50609011(CHEMBL5287921)
Affinity DataKi:  1.27E+3nMAssay Description:Displacement of [125]IBNtxA from mouse KOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Memorial Sloan Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50531606(CHEMBL4514672)
Affinity DataKi:  1.28E+3nMAssay Description:Displacement of [3H]N-methylspiperone from human D4 receptor by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Memorial Sloan Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50531605(CHEMBL4552298)
Affinity DataKi:  1.63E+3nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)TBA
LigandPNGBDBM50609011(CHEMBL5287921)
Affinity DataKi:  1.68E+3nMAssay Description:Displacement of [125]IBNtxA from mouse MOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Memorial Sloan Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50531606(CHEMBL4514672)
Affinity DataKi:  1.71E+3nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50474151(CHEMBL292521)
Affinity DataKi:  1.88E+3nMAssay Description:Displacement of [125]IBNtxA from mouse DOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Memorial Sloan Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50531605(CHEMBL4552298)
Affinity DataKi:  2.05E+3nMAssay Description:Displacement of [3H]LSD from human 5-HT2B receptor expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Mus musculus (Mouse))TBA
LigandPNGBDBM50566316(CHEMBL4859858)
Affinity DataKi:  2.20E+3nMAssay Description:Displacement of [125]IBNtxA from mouse KOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Memorial Sloan Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50531606(CHEMBL4514672)
Affinity DataKi:  2.56E+3nMAssay Description:Displacement of [3H]WIN35428 from human DAT receptor expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Memorial Sloan Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50531606(CHEMBL4514672)
Affinity DataKi:  2.77E+3nMAssay Description:Displacement of [3H]LSD from human 5-HT7 receptor expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50609011(CHEMBL5287921)
Affinity DataKi:  3.24E+3nMAssay Description:Displacement of [125]IBNtxA from mouse DOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Memorial Sloan Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50531606(CHEMBL4514672)
Affinity DataKi:  3.36E+3nMAssay Description:Displacement of [3H] NECA from human adrenergic alpha 2A receptor expressed in MDCK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50566317(CHEMBL4848517)
Affinity DataKi:  3.40E+3nMAssay Description:Displacement of [125]IBNtxA from mouse DOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50609009(CHEMBL56717)
Affinity DataKi:  4.14E+3nMAssay Description:Displacement of [125]IBNtxA from mouse DOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMu-type opioid receptor(MOUSE)TBA
LigandPNGBDBM50609009(CHEMBL56717)
Affinity DataKi:  6.90E+3nMAssay Description:Displacement of [125]IBNtxA from mouse MOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKappa-type opioid receptor(Mus musculus (Mouse))TBA
LigandPNGBDBM50609009(CHEMBL56717)
Affinity DataKi:  7.18E+3nMAssay Description:Displacement of [125]IBNtxA from mouse KOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50566316(CHEMBL4859858)
Affinity DataKi:  7.95E+3nMAssay Description:Displacement of [125]IBNtxA from mouse DOR stably expressed in CHO cell membranes incubated for 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Memorial Sloan Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50531607(CHEMBL4472251)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50609010(CHEMBL5276728)
Affinity DataIC50:  1.10E+3nMAssay Description:Antagonist activity at mouse DOR expressed in CHO cell membranes assessed as inhibition of DPDPE induced [35S]-GTPgammaS binding incubated for 60 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50566317(CHEMBL4848517)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at mouse DOR expressed in CHO cell membranes assessed as inhibition of DPDPE induced [35S]-GTPgammaS binding incubated for 60 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMu-type opioid receptor(MOUSE)TBA
LigandPNGBDBM50519927(CHEMBL4546925)
Affinity DataIC50:  1.09E+4nMAssay Description:Antagonist activity at mouse MOR expressed in CHO cell membranes assessed as inhibition of DAMGO induced [35S]-GTPgammaS binding incubated for 60 min...More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50519927(CHEMBL4546925)
Affinity DataIC50:  1.26E+4nMAssay Description:Antagonist activity at mouse DOR expressed in CHO cell membranes assessed as inhibition of DPDPE induced [35S]-GTPgammaS binding incubated for 60 min...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Memorial Sloan Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50554763(CHEMBL4758061)
Affinity DataEC50:  83nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human MOR expressed in human U2OS cell membranes assessed as stimulation of [35S]-GTPgammaS bind...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Memorial Sloan Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50554764(CHEMBL4761310)
Affinity DataEC50:  110nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human MOR expressed in human U2OS cell membranes assessed as stimulation of [35S]-GTPgammaS bind...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Memorial Sloan Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50554765(CHEMBL4781906)
Affinity DataEC50:  205nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human MOR expressed in human U2OS cell membranes assessed as stimulation of [35S]-GTPgammaS bind...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Memorial Sloan Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50554766(CHEMBL4795492)
Affinity DataEC50:  0.400nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human MOR expressed in human U2OS cell membranes assessed as stimulation of [35S]-GTPgammaS bind...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Memorial Sloan Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50554767(CHEMBL4776176)
Affinity DataEC50:  144nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human MOR expressed in human U2OS cell membranes assessed as stimulation of [35S]-GTPgammaS bind...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Memorial Sloan Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50554768(CHEMBL4783765)
Affinity DataEC50:  85nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human MOR expressed in human U2OS cell membranes assessed as stimulation of [35S]-GTPgammaS bind...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Memorial Sloan Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50554769(CHEMBL4788377)
Affinity DataEC50:  32nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human MOR expressed in human U2OS cell membranes assessed as stimulation of [35S]-GTPgammaS bind...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Memorial Sloan Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50554770(CHEMBL4783653)
Affinity DataEC50:  163nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human MOR expressed in human U2OS cell membranes assessed as stimulation of [35S]-GTPgammaS bind...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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